SCHEMBL13765699

SCHEMBL13765699

CNc1cc(OCCOC)c(OC)cc1C(=N)N1CCN(C(=O)Nc2ccc(Oc3ccccc3)cc2)CC1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 20/20 0.61
KIT P10721 1/20 0.51
FGFR1 P11362 1/20 0.51
PDGFRA P16234 1/20 0.51
FGFR2 P21802 1/20 0.51
FGFR4 P22455 1/20 0.51
FGFR3 P22607 1/20 0.51
FLT3 P36888 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13360884 0.94 PDGFRB (0.59) PDGFRBKITFGFR1PDGFRAFGFR2
SCHEMBL13360876 0.87 PDGFRB (0.66) PDGFRBKITFLT3
SCHEMBL13105997 0.78 PDGFRB (0.64) PDGFRBKITFGFR1PDGFRAFGFR2
SCHEMBL13330456 0.76 PDGFRB (1.00) PDGFRBKITFGFR1PDGFRAFGFR2
SCHEMBL13360952 0.76 PDGFRB (0.52) PDGFRBKITFGFR1PDGFRAFGFR2
SCHEMBL13330467 0.70 PDGFRB (0.95) PDGFRBKITFGFR1PDGFRAFGFR2
SCHEMBL13330468 0.69 PDGFRB (0.88) PDGFRBKITFGFR1PDGFRAFGFR2
SCHEMBL13773428 0.68 PDGFRB (0.58) PDGFRBKITFGFR1PDGFRAFGFR2
SCHEMBL13932716 0.68 SRC (0.39) FGFR1FGFR2FGFR4FGFR3
SCHEMBL2592017 0.67 PDGFRB (1.00) PDGFRBKITFGFR1PDGFRAFGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7560461-B2 Quinazoline derivatives as kinase inhibitors MILLENNIUM PHARMACEUTICALS, INC. (US) 2009-07-14 US disclosed