SCHEMBL13765757

SCHEMBL13765757

Cc1cc(F)ccc1-c1nc(Cl)nc2[nH]cnc12

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 6/20 0.48
GRIN1 Q05586 2/20 0.34
GRIN2B Q13224 2/20 0.34
RXFP1 Q9HBX9 1/20 0.33
PLK4 O00444 1/20 0.33
PAK4 O96013 1/20 0.33
XDH P47989 1/20 0.33
CTSA P10619 1/20 0.32
ABL1 P00519 1/20 0.32
MAPK14 Q16539 1/20 0.31
SLC34A1 Q06495 1/20 0.31
GRM5 P41594 1/20 0.31
PIK3CA P42336 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13765756 0.86 HSP90AB1 (0.50) HSP90AB1XDHABL1
SCHEMBL13765750 0.86 HSP90AB1 (0.40) HSP90AB1PLK4PAK4XDH
SCHEMBL4090407 0.82 HSP90AB1 (0.68) HSP90AB1GRIN1GRIN2BRXFP1
SCHEMBL13765755 0.80 KDM4E (0.35) HSP90AB1PLK4PAK4XDH
SCHEMBL13765751 0.78 PARP1 (0.36) HSP90AB1PAK4XDHABL1MAPK14
SCHEMBL4089680 0.76 DPP4 (0.46) HSP90AB1PIK3CA
SCHEMBL14249312 0.75 HSP90AB1 (0.43) HSP90AB1MAPK14
SCHEMBL24010622 0.75 HSP90AB1 (0.39) HSP90AB1CTSAMAPK14GRM5
SCHEMBL30160025 0.75 HSP90AB1 (0.39) HSP90AB1CTSAMAPK14GRM5
SCHEMBL4259002 0.75 XDH (0.32) HSP90AB1XDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090181989-A1 Purine Compunds as HSP90 Protein Inhibitors for the Treatment of Cancer VERNALIS ( R & D) LTD. (GB) 2009-07-16 US disclosed
US-20090181989-A1 Purine Compunds as HSP90 Protein Inhibitors for the Treatment of Cancer VERNALIS ( R & D) LTD. (GB) 2009-07-16 US disclosed
WO-2007034185-A1 PURINE COMPOUNDS AS HSP90 PROTEIN INHIBITORS FOR THE TREATMENT OF CANCER VERNALIS (R & D) LTD. (GB) 2007-03-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090181989-A1 Purine Compunds as HSP90 Protein Inhibitors for the Treatment of Cancer HSP90AA1, HSP90AB1, HSP90AB2P HSP90AB1 2/4885GRIN1 4086/4885GRIN2B 4287/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.