SCHEMBL13769142

SCHEMBL13769142

Cc1ccc2c(N3CCCCC3)nc(-c3ccccc3O)nc2c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMAD3 P84022 1/20 0.71
KMT2A Q03164 4/20 0.60
MEN1 O00255 2/20 0.60
ALDH1A1 P00352 5/20 0.57
TSHR P16473 5/20 0.57
HSD17B10 Q99714 3/20 0.57
KDM4E B2RXH2 3/20 0.57
MAPK1 P28482 3/20 0.57
HPGD P15428 2/20 0.57
LMNA P02545 2/20 0.57
TDP1 Q9NUW8 2/20 0.57
USP2 O75604 2/20 0.57
NPSR1 Q6W5P4 1/20 0.57
HIF1A Q16665 2/20 0.54
L3MBTL1 Q9Y468 3/20 0.53
MAPT P10636 2/20 0.53
ABCB1 P08183 1/20 0.51
CHEK2 O96017 1/20 0.50
ACP1 P24666 2/20 0.49
METAP1 P53582 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2734047 0.99 SMAD3 (0.73) SMAD3KMT2AMEN1ALDH1A1TSHR
SCHEMBL1084601 0.91 SMAD3 (0.71) SMAD3KMT2AMEN1ALDH1A1TSHR
SCHEMBL1084032 0.90 MEN1 (0.70) SMAD3KMT2AMEN1ALDH1A1TSHR
SCHEMBL1084599 0.90 SMAD3 (0.57) SMAD3KMT2AMEN1ALDH1A1TSHR
SCHEMBL13769477 0.89 MEN1 (0.76) SMAD3KMT2AMEN1ALDH1A1TSHR
SCHEMBL5506324 0.89 SMAD3 (0.62) SMAD3KMT2AMEN1ALDH1A1TSHR
SCHEMBL1084790 0.88 SMAD3 (0.58) SMAD3KMT2AMEN1ALDH1A1TSHR
SCHEMBL295770 0.88 CYP1A2 (0.61) SMAD3KMT2AMEN1ALDH1A1TSHR
SCHEMBL1084946 0.88 CYP1A2 (0.61) SMAD3KMT2AMEN1ALDH1A1TSHR
SCHEMBL1084859 0.88 SMAD3 (0.58) SMAD3KMT2AMEN1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784393-B1 QUINAZOLINES USEFUL AS MODULATORS OF ION CHANNELS VERTEX PHARMA (US) 2009-07-01 EP disclosed