SCHEMBL13769780

SCHEMBL13769780

CC1C=CC(Cn2cc(C(=O)Nc3c[nH]c(=O)c(-c4cc5cc(CNCCO)ccc5[nH]4)c3)cn2)=CC1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 10/20 0.35
RPS6KA3 P51812 4/20 0.33
RPS6KA2 Q15349 3/20 0.33
RPS6KA1 Q15418 3/20 0.33
RPS6KA6 Q9UK32 3/20 0.33
KLKB1 P03952 4/20 0.32
BUB1 O43683 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13769995 0.89 CHEK1 (0.46) CHEK1
SCHEMBL13769772 0.88 CHEK1 (0.40) CHEK1RPS6KA3RPS6KA2RPS6KA1RPS6KA6
SCHEMBL13770126 0.88 CHEK1 (0.42) CHEK1
SCHEMBL13770146 0.87 CHEK1 (0.47) CHEK1
SCHEMBL13770383 0.87 RPS6KA2 (0.38) RPS6KA3RPS6KA2RPS6KA1RPS6KA6BUB1
SCHEMBL13770409 0.87 CHEK1 (0.36) CHEK1RPS6KA3RPS6KA2RPS6KA1RPS6KA6
SCHEMBL951161 0.85 KLKB1 (0.41) CHEK1RPS6KA3RPS6KA2RPS6KA1RPS6KA6
SCHEMBL13770545 0.85 KDR (0.36) CHEK1RPS6KA3RPS6KA2RPS6KA1RPS6KA6
SCHEMBL950328 0.85 SMN1; SMN2 (0.39) CHEK1KLKB1
SCHEMBL950208 0.85 RPS6KA3 (0.40) RPS6KA3RPS6KA2RPS6KA1RPS6KA6KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009093012-A1 INDOLYL- PYRIDONE DERIVATIVES HAVING CHECKPOINT KINASE 1 INHIBITORY ACTIVITY VERNALIS (R & D) LTD (GB) 2009-07-30 WO disclosed