SCHEMBL1377159

SCHEMBL1377159

Cc1nc(NC(=O)c2cnn3c(C(F)(F)F)cc(-c4ccc(C(F)(F)F)c(Cl)c4)nc23)sc1S(N)(=O)=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 9/20 0.47
TSHR P16473 6/20 0.47
MAPK1 P28482 4/20 0.47
NPSR1 Q6W5P4 4/20 0.47
MAPT P10636 3/20 0.47
USP2 O75604 1/20 0.47
PKM P14618 1/20 0.47
KDM4E B2RXH2 10/20 0.47
ALDH1A1 P00352 8/20 0.46
POLB P06746 4/20 0.46
THRB P10828 1/20 0.46
HPGD P15428 6/20 0.45
CASP1 P29466 4/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
LMNA P02545 3/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HTT P42858 2/20 0.42
CASP7 P55210 3/20 0.42
GLA P06280 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1939254 0.94 HSD17B10 (0.49) HSD17B10TSHRMAPK1NPSR1MAPT
SCHEMBL1381357 0.92 HSD17B10 (0.49) HSD17B10TSHRMAPK1NPSR1MAPT
SCHEMBL1378159 0.91 HSD17B10 (0.54) HSD17B10TSHRMAPK1NPSR1MAPT
SCHEMBL1939111 0.89 KDM4E (0.44) HSD17B10TSHRMAPK1NPSR1MAPT
SCHEMBL1938554 0.88 THRB (0.51) HSD17B10TSHRMAPK1NPSR1MAPT
SCHEMBL1382183 0.88 KDM4E (0.53) HSD17B10TSHRMAPK1NPSR1MAPT
SCHEMBL1939595 0.88 THRB (0.52) HSD17B10TSHRMAPK1NPSR1MAPT
SCHEMBL1940392 0.87 KDM4E (0.41) HSD17B10TSHRMAPK1NPSR1MAPT
SCHEMBL1939384 0.83 KMT2A (0.50) HSD17B10MAPK1NPSR1MAPTKDM4E
SCHEMBL1939421 0.82 KDM4E (0.45) HSD17B10TSHRMAPK1NPSR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4708438-B2 2011-06-22 JP claimed
EP-1851225-B1 PYRAZOLO-PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2011-06-15 EP claimed
EP-1851225-B1 PYRAZOLO-PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2011-06-15 EP disclosed