SCHEMBL1377595

SCHEMBL1377595

N#CCNC(=O)[C@@H]1CCCCC1c1ccccc1-c1cccc(N)c1

nearest known ligand 0.67

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSK P43235 18/20 0.67
CTSL P07711 2/20 0.45
CTSB P07858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4983624 1.00 CTSK (0.67) CTSKCTSLCTSB
SCHEMBL1379169 0.89 CTSK (0.68) CTSKCTSLCTSB
SCHEMBL4990609 0.89 CTSK (0.68) CTSKCTSLCTSB
SCHEMBL5685690 0.88 CTSK (0.67) CTSKCTSLCTSB
SCHEMBL4984927 0.88 CTSK (0.67) CTSKCTSLCTSB
SCHEMBL1378911 0.88 CTSK (0.67) CTSKCTSLCTSB
SCHEMBL4988700 0.87 CTSK (0.69) CTSKCTSLCTSB
SCHEMBL1378507 0.87 CTSK (0.66) CTSKCTSLCTSB
SCHEMBL4986683 0.87 CTSK (0.66) CTSKCTSLCTSB
SCHEMBL4991669 0.86 CTSK (0.65) CTSKCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4690319-B2 2011-06-01 JP claimed
EP-1644326-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS Merck Frosst Canada Ltd. (CA) 2006-04-12 EP claimed
WO-2005000800-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD. (CA) 2005-01-06 WO claimed