SCHEMBL1378096

SCHEMBL1378096

CCC(CC)Nc1nc(NCc2cccnc2)c2ncn(C(C)C)c2n1

nearest known ligand 0.89

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 20/20 0.89
CDK1 P06493 17/20 0.89
CDK7 P50613 17/20 0.89
CDK4 P11802 15/20 0.89
CCNE1 P24864 15/20 0.89
MAPK1 P28482 14/20 0.89
CCNH P51946 14/20 0.89
CCNB1 P14635 13/20 0.89
CCND1 P24385 13/20 0.89
CDK9 P50750 10/20 0.80
CCNT1 O60563 5/20 0.80
CDK5 Q00535 4/20 0.80
MNAT1 P51948 2/20 0.80
CDK6 Q00534 2/20 0.80
CSNK1D P48730 2/20 0.71
CLK2 P49760 2/20 0.71
CSNK1G2 P78368 2/20 0.71
DYRK1A Q13627 2/20 0.71
CLK4 Q9HAZ1 2/20 0.71
CSNK1G1 Q9HCP0 2/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17628584 0.94 CDK2 (1.00) CDK2CDK1CDK7CDK4CCNE1
SCHEMBL1375655 0.94 CDK2 (0.83) CDK2CDK1CDK7CDK4CCNE1
SCHEMBL1378255 0.94 CDK2 (0.83) CDK2CDK1CDK7CDK4CCNE1
SCHEMBL13633363 0.94 CDK2 (1.00) CDK2CDK1CDK7CDK4CCNE1
SCHEMBL3749485 0.90 CDK2 (0.86) CDK2CDK1CDK7CDK4CCNE1
SCHEMBL14403894 0.89 CDK1 (0.88) CDK2CDK1CDK7CDK4CCNE1
SCHEMBL29829223 0.89 CDK2 (1.00) CDK2CDK1CDK7CDK4CCNE1
SCHEMBL1378920 0.89 CDK2 (1.00) CDK2CDK1CDK7CDK4CCNE1
SCHEMBL1374884 0.89 CDK2 (1.00) CDK2CDK1CDK7CDK4CCNE1
SCHEMBL3336119 0.89 CDK2 (1.00) CDK2CDK1CDK7CDK4CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4723858-B2 2011-07-13 JP claimed
JP-2006506341-A 2006-02-23 JP claimed
EP-1529047-A2 NEW PURINE DERIVATIVES Cyclacel Limited (GB) 2005-05-11 EP claimed
WO-2004016612-A2 NEW PURINE DERIVATIVES CYCLACEL LIMITED (GB) 2004-02-26 WO claimed
EP-1951307-A2 COMBINATION OF A CDK-INHIBITOR AND A HDAC-INHIBITOR Cyclacel Limited (GB) 2008-08-06 EP disclosed
WO-2007054725-A2 COMBINATION OF A CDK-INHIBITOR AND A HDAC-INHIBITOR CYCLACEL LIMITED (GB) 2007-05-18 WO disclosed
EP-1529047-A2 NEW PURINE DERIVATIVES Cyclacel Limited (GB) 2005-05-11 EP disclosed
WO-2004016612-A2 NEW PURINE DERIVATIVES CYCLACEL LIMITED (GB) 2004-02-26 WO disclosed