SCHEMBL13786191

SCHEMBL13786191

CCC(CI)(c1ccc(OCC(O)C(C)(C)C)c(C)c1)c1cc(C)c(CN(CC(=O)N=O)C(C)=O)s1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 9/20 0.55
HDAC3 O15379 5/20 0.55
HDAC1 Q13547 1/20 0.46
VDR P11473 9/20 0.45
AR P10275 4/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3391016 0.86 HDAC6 (0.63) HDAC6HDAC3HDAC1VDRAR
SCHEMBL13786339 0.77 HDAC6 (0.69) HDAC6HDAC3HDAC1VDRAR
SCHEMBL13672879 0.75 HDAC6 (0.72) HDAC6HDAC3HDAC1VDRAR
SCHEMBL13949123 0.74 HDAC6 (0.60) HDAC6HDAC3HDAC1VDRAR
SCHEMBL3394923 0.74 HDAC6 (0.71) HDAC6HDAC3HDAC1VDRAR
SCHEMBL13366691 0.73 HDAC6 (0.81) HDAC6HDAC3HDAC1VDRAR
SCHEMBL3391135 0.73 HDAC6 (0.69) HDAC6HDAC3HDAC1VDRAR
SCHEMBL13786026 0.73 HDAC6 (0.66) HDAC6HDAC3HDAC1VDRAR
SCHEMBL13786239 0.73 HDAC6 (0.59) HDAC6HDAC3HDAC1VDRAR
SCHEMBL3388896 0.72 VDR (0.57) HDAC6HDAC3VDRAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1511740-B1 PHENYL-THIOPHENE TYPE VITAMIN D RECEPTOR MODULATORS LILLY CO ELI (US) 2009-07-08 EP disclosed