SCHEMBL13786309

SCHEMBL13786309

CCc1cc(C(CC)(CC)c2ccc(C(=O)O)s2)ccc1CCC(N=O)C(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.36
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
ATM Q13315 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
HDAC3 O15379 2/20 0.33
GRIN2C Q14957 1/20 0.32
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13785988 0.87 HDAC3 (0.31) HPGDTSHRMAPK1ATMNPSR1
SCHEMBL13786141 0.83 DAO (0.36) DAOHPGDTSHRMAPK1ATM
SCHEMBL13786075 0.78 HDAC3 (0.39) HDAC3HDAC6
SCHEMBL13786179 0.78 HDAC6 (0.47) HDAC3HDAC6
SCHEMBL13786294 0.75 HDAC3 (0.42) DAOHPGDTSHRMAPK1ATM
SCHEMBL13786250 0.74 DAO (0.38) DAOHPGDTSHRMAPK1ATM
SCHEMBL13785989 0.74 ESR1 (0.33) HPGDTSHRMAPK1ATMNPSR1
SCHEMBL13786182 0.73 NPSR1 (0.48) HPGDTSHRMAPK1ATMNPSR1
SCHEMBL3396321 0.73 HDAC6 (0.50) HDAC3HDAC6
SCHEMBL13785975 0.72 HDAC3 (0.47) NPSR1HDAC3HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1511740-B1 PHENYL-THIOPHENE TYPE VITAMIN D RECEPTOR MODULATORS LILLY CO ELI (US) 2009-07-08 EP disclosed