SCHEMBL1379088

SCHEMBL1379088

CC(C)(C)CCNc1n[nH]c2c(F)c(Cl)c(-c3ccccc3)cc12.Fc1c(Cl)c(-c2ccccc2)cc2c(NCCCc3ccccc3)n[nH]c12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.53
CDK1 P06493 2/20 0.53
CDK2 P24941 2/20 0.53
PIK3CD O00329 2/20 0.37
PIK3R1 P27986 1/20 0.37
CDC7 O00311 1/20 0.34
TYMP P19971 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
GBA1 P04062 1/20 0.33
TP53 P04637 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.32
FGFR1 P11362 1/20 0.32
ADK P55263 1/20 0.32
FFAR1 O14842 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2338648 0.92 GSK3B (0.58) GSK3BCDK1CDK2PIK3CDPIK3R1
SCHEMBL2335996 0.92 GSK3B (0.60) GSK3BCDK1CDK2CDC7CYP1A2
SCHEMBL2337764 0.86 GSK3B (0.60) GSK3BCDK1CDK2LMNATP53
SCHEMBL6528308 0.84 GSK3B (0.50) GSK3BCDK1CDK2PIK3CDPIK3R1
SCHEMBL2337774 0.83 GSK3B (0.57) GSK3BCDK1CDK2CDC7FGFR1
SCHEMBL2338246 0.83 GSK3B (0.59) GSK3BCDK1CDK2CDC7FGFR1
SCHEMBL2333642 0.83 GSK3B (0.67) GSK3BCDK1CDK2CDC7CYP1A2
SCHEMBL1375621 0.82 GSK3B (0.64) GSK3BCDK1CDK2CDC7LMNA
SCHEMBL1378947 0.81 GSK3B (0.70) GSK3BCDK1CDK2CDC7CYP1A2
SCHEMBL1375627 0.81 GSK3B (0.58) GSK3BCDK1CDK2CDC7CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4764168-B2 2011-08-31 JP claimed
EP-1572200-A1 AMINOINDAZOLE DERIVATIVES AND USE THEREOF AS KINASE INHIBITORS Aventis Pharma S.A. (FR) 2005-09-14 EP claimed
WO-2004062662-A1 AMINOINDAZOLE DERIVATIVES AND USE THEREOF AS KINASE INHIBITORS AVENTIS PHARMA S.A. (FR) 2004-07-29 WO claimed