SCHEMBL13804384

SCHEMBL13804384

CN1CCC[C@@H](c2nnn[nH]2)C1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.39
KCNH2 Q12809 4/20 0.36
HTR2A P28223 3/20 0.36
DRD2 P14416 2/20 0.36
HTR2C P28335 1/20 0.36
MAPK11 Q15759 1/20 0.36
MAPK14 Q16539 1/20 0.36
ERCC1 P07992 1/20 0.36
ERCC4 Q92889 1/20 0.36
DRD3 P35462 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
LSS P48449 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12853575 0.82
SCHEMBL12258869 0.80 PARP1 (0.42) PARP1KCNH2DRD2DRD3
SCHEMBL9910973 0.79 DRD4 (0.35) PARP1HTR2AMAPK11MAPK14ERCC1
SCHEMBL6199606 0.77 POLB (0.31) DRD2DRD3
SCHEMBL7856962 0.76
SCHEMBL2335166 0.76 ALDH1A1 (0.38)
SCHEMBL10407882 0.74 OPRL1 (0.38) PARP1DRD2DRD3
SCHEMBL7853880 0.74 ALDH1A1 (0.41)
SCHEMBL7852075 0.74 ALDH1A1 (0.41)
SCHEMBL10407881 0.73 PARP1 (0.40) PARP1DRD2ERCC1ERCC4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225238-B1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZOÝ1,2- ¨IMIDAZOLE-3- CARBOXYLIC ACID AMIDES BOEHRINGER INGELHEIM INT (DE) 2014-09-03 EP disclosed
WO-2009070485-A1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZO[1,2-α]IMIDAZOLE-3- CARBOXYLIC ACID AMIDES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-06-04 WO disclosed