SCHEMBL1380840

SCHEMBL1380840

CO[C@@H](N)CC[C@H]1CN(c2c(F)cc3c(=O)n(N)c(=O)n(C4CC4)c3c2C)C[C@@H]1C

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 10/20 0.38
SCN5A Q14524 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
CACNA1C Q13936 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7515541 0.91 KCNH2 (0.38) KCNH2
SCHEMBL1382756 0.86 KCNH2 (0.38) KCNH2SCN5A
SCHEMBL7552000 0.86 KCNH2 (0.40) KCNH2SCN5ACYP1A2CYP3A4CYP2D6
SCHEMBL1382759 0.86 KCNH2 (0.38) KCNH2SCN5A
SCHEMBL1382762 0.86 KCNH2 (0.38) KCNH2SCN5A
Hydrochloric Acid SCHEMBL4512757 0.86 KCNH2 (0.37) KCNH2SCN5A
Hydrochloric Acid SCHEMBL4512744 0.86 KCNH2 (0.37) KCNH2SCN5A
Hydrochloric Acid SCHEMBL4512749 0.86 KCNH2 (0.37) KCNH2SCN5A
SCHEMBL1380249 0.84 KCNH2 (0.37) KCNH2SCN5ACYP1A2CYP3A4CYP2D6
SCHEMBL4526634 0.83 KCNH2 (0.38) KCNH2SCN5ACYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4811978-B2 2011-11-09 JP claimed
EP-1255739-A1 3-AMINOQUINAZOLIN-2,4-DIONE ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 2002-11-13 EP claimed
WO-2001053273-A1 3-AMINOQUINAZOLIN-2,4-DIONE ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 2001-07-26 WO claimed
EP-1255739-A1 3-AMINOQUINAZOLIN-2,4-DIONE ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 2002-11-13 EP disclosed
WO-2001053273-A1 3-AMINOQUINAZOLIN-2,4-DIONE ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 2001-07-26 WO disclosed