SCHEMBL1380843

SCHEMBL1380843

O[C@@H](COc1ccc(-c2onc3cc(F)ccc23)cc1)CN1CCC(O)(c2ccccc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 11/20 0.48
PKM P14618 1/20 0.46
HTR2A P28223 2/20 0.42
HTR1A P08908 1/20 0.42
DRD2 P14416 1/20 0.42
CHRNA7 P36544 1/20 0.42
ALDH1A1 P00352 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ADRB3 P13945 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7489075 1.00 ABCB1 (0.48) ABCB1PKMHTR2AHTR1ADRD2
SCHEMBL1383560 0.86 MAPT (0.55) ABCB1ALDH1A1L3MBTL1
SCHEMBL1383563 0.86 MAPT (0.55) ABCB1ALDH1A1L3MBTL1
SCHEMBL5374878 0.86 HTR2A (0.49) ABCB1PKMHTR2AHTR1ADRD2
SCHEMBL5366093 0.86 HTR2A (0.49) ABCB1PKMHTR2AHTR1ADRD2
SCHEMBL5366098 0.86 HTR2A (0.49) ABCB1PKMHTR2AHTR1ADRD2
SCHEMBL7500542 0.85 HTR2A (0.51) PKMHTR2AHTR1ADRD2CHRNA7
SCHEMBL7497905 0.85 HTR2A (0.51) PKMHTR2AHTR1ADRD2CHRNA7
SCHEMBL16808047 0.82 ABCB1 (0.63) ABCB1L3MBTL1
SCHEMBL16808048 0.82 ABCB1 (0.63) ABCB1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4806149-B2 2011-11-02 JP claimed
EP-1216244-A1 Benzisoxazolyl-, pyridoisoxazolyl- and benzthienyl-phenoxy derivatives useful as D4 antagonists Aventis Pharmaceuticals Inc. (US) 2002-06-26 EP claimed
WO-2001019821-A1 BENZISOXAZOLYL-, PYRIDOISOXAZOLYL- AND BENZTHIENYL-PHENOXY DERIVATIVES USEFUL AS D4 ANTAGONISTS AVENTIS PHARMACEUTICALS INC. (US) 2001-03-22 WO claimed
EP-1216244-A1 Benzisoxazolyl-, pyridoisoxazolyl- and benzthienyl-phenoxy derivatives useful as D4 antagonists Aventis Pharmaceuticals Inc. (US) 2002-06-26 EP disclosed
WO-2001019821-A1 BENZISOXAZOLYL-, PYRIDOISOXAZOLYL- AND BENZTHIENYL-PHENOXY DERIVATIVES USEFUL AS D4 ANTAGONISTS AVENTIS PHARMACEUTICALS INC. (US) 2001-03-22 WO disclosed