SCHEMBL1380933

SCHEMBL1380933

NC(=O)C=Cc1ccoc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.69
MAPT P10636 4/20 0.54
ALOX5 P09917 3/20 0.54
ALDH1A1 P00352 3/20 0.54
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
KMT2A Q03164 4/20 0.43
POLB P06746 4/20 0.43
MEN1 O00255 3/20 0.43
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.43
LMNA P02545 1/20 0.43
PKM P14618 1/20 0.43
HTT P42858 1/20 0.43
BLM P54132 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CYP1A2 P05177 3/20 0.41
CYP2C19 P33261 2/20 0.41
CYP1A1 P04798 1/20 0.41
CYP1B1 Q16678 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2815054 1.00 HCAR2 (0.69) HCAR2MAPTALOX5ALDH1A1MAOA
SCHEMBL7893859 0.82 HCAR2 (1.00) HCAR2MAPTALOX5ALDH1A1MAOA
SCHEMBL660178 0.82 HCAR2 (1.00) HCAR2MAPTALOX5ALDH1A1MAOA
SCHEMBL564789 0.82 HCAR2 (1.00) HCAR2MAPTALOX5ALDH1A1MAOA
SCHEMBL28981304 0.80 HCAR2 (0.69) HCAR2MAPTALOX5ALDH1A1MAOA
SCHEMBL3513899 0.80 HCAR2 (0.69) HCAR2MAPTALOX5ALDH1A1MAOA
SCHEMBL6832853 0.80 HCAR2 (0.69) HCAR2MAPTALOX5ALDH1A1MAOA
Hydrochloric Acid SCHEMBL9261463 0.80 HCAR2 (0.96) HCAR2MAPTALOX5ALDH1A1MAOA
SCHEMBL13692335 0.80 HCAR2 (0.69) HCAR2MAPTALOX5ALDH1A1MAOA
SCHEMBL14504206 0.78 HCAR2 (0.56) HCAR2MAPTALOX5ALDH1A1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4828407-B2 2011-11-30 JP claimed
EP-1594869-A2 3-SUBSTITUTED-2(ARYLALKYL)-1-AZABICYCLOALKANES AND METHODS OF USE THEREOF Targacept, Inc. (US) 2005-11-16 EP claimed
WO-2004076449-A2 3-SUBSTITUTED-2(ARYLALKYL)-1-AZABICYCLOALKANES AND METHODS OF USE THEREOF TARGACEPT, INC. (US) 2004-09-10 WO claimed
US-20100247938-A1 MATERIAL FOR THREE-DIMENSIONAL MODELING, PROCESS FOR PRODUCING THREE-DIMENSIONAL MODEL, AND THREE-DIMENSIONAL MODEL FUJIFILM CORPORATION (JP) 2010-09-30 US disclosed