SCHEMBL13811482

SCHEMBL13811482

Cc1cc(I)ccc1OCC(=O)Nc1ccc(OCC=O)c(Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.53
NFKB1 P19838 2/20 0.53
RAB9A P51151 2/20 0.53
NFKB2 Q00653 2/20 0.53
RELA Q04206 2/20 0.53
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
ALDH1A1 P00352 4/20 0.47
POLB P06746 2/20 0.47
HPGD P15428 2/20 0.46
MAPT P10636 3/20 0.46
HTT P42858 2/20 0.46
GBA1 P04062 1/20 0.46
LMNA P02545 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
TP53 P04637 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4014301 0.83 MEN1 (0.67) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL4007988 0.82 KDR (0.52) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL4015603 0.78 NPC1 (0.49) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL16063220 0.72 NPC1 (0.65) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL31258533 0.70 MEN1 (0.58) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL31258534 0.70 MEN1 (0.58) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL10857636 0.69 NOTUM (0.70) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL11475652 0.69 SMN1; SMN2 (0.69) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL12259122 0.69 L3MBTL1 (0.64) NPC1MEN1KMT2APOLBMAPT
SCHEMBL10144037 0.69 KDM4E (0.50) NPC1MEN1KMT2AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558567-B1 NOVEL AMIDE COMPOUNDS WITH MCH ANTAGONISTIC EFFECT AND MEDICAMENTS COMPRISING SAID COMPOUNDS BOEHRINGER INGELHEIM PHARMA (DE) 2009-06-24 EP disclosed
US-7351719-B2 Amide compounds having MCH-antagonistic activity and medicaments comprising these compounds BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2008-04-01 US disclosed
US-7351719-B2 Amide compounds having MCH-antagonistic activity and medicaments comprising these compounds BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2008-04-01 US disclosed