SCHEMBL13818145

SCHEMBL13818145

C[C@@H]1C(=O)N(C(=O)OC(C)(C)C)CC[C@H]1c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.45
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
GPR119 Q8TDV5 1/20 0.44
KDM1A O60341 2/20 0.43
TACR1 P25103 1/20 0.42
MAOB P27338 1/20 0.41
STS P08842 1/20 0.41
KDM4E B2RXH2 1/20 0.40
PKM P14618 1/20 0.40
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 2/20 0.40
SLC6A3 Q01959 2/20 0.40
HRH3 Q9Y5N1 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ABCB1 P08183 1/20 0.39
RIPK1 Q13546 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18252865 0.87 GPR119 (0.47) PDE4APDE4BPDE4CPDE4DGPR119
SCHEMBL31510733 0.86 PDE4A (0.49) PDE4APDE4BPDE4CPDE4DGPR119
SCHEMBL18255018 0.83 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DSTS
SCHEMBL18247835 0.83 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DSTS
SCHEMBL3730368 0.83 PDE4A (0.57) RORCPDE4APDE4BPDE4CPDE4D
SCHEMBL18245067 0.81 ATM (0.43) PDE4APDE4BPDE4CPDE4DMEN1
SCHEMBL18244795 0.81 ATM (0.43) PDE4APDE4BPDE4CPDE4DMEN1
SCHEMBL3163882 0.81 ATM (0.43) PDE4APDE4BPDE4CPDE4DMEN1
SCHEMBL31510707 0.79 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DGPR119
SCHEMBL24433813 0.79 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7553841-B2 Amino cyclobutylamide modulators of chemokine receptor activity MERCK & CO., INC. (US) 2009-06-30 US disclosed