SCHEMBL13822838

SCHEMBL13822838

Nc1ccccc1NC(=O)c1nc2c(s1)CN(C(=O)Nc1ccc(C(=O)O)cc1)CC2

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 4/20 0.51
HDAC1 Q13547 3/20 0.51
HDAC6 Q9UBN7 2/20 0.51
F10 P00742 15/20 0.47
F11 P03951 1/20 0.46
HDAC2 Q92769 1/20 0.42
NCOR2 Q9Y618 1/20 0.42
PIK3CA P42336 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL977976 0.93 HDAC3 (0.51) HDAC3HDAC1HDAC6F10HDAC2
SCHEMBL978289 0.90 HDAC3 (0.47) HDAC3HDAC1HDAC6F10PIK3CA
SCHEMBL975313 0.90 F10 (0.51) HDAC3HDAC1HDAC6F10HDAC2
SCHEMBL13822776 0.90 HDAC3 (0.56) HDAC3HDAC1HDAC6F10F11
SCHEMBL978994 0.89 F10 (0.47) HDAC3HDAC1HDAC6F10
SCHEMBL977872 0.89 HDAC3 (0.45) HDAC3HDAC1HDAC6F10
SCHEMBL13822915 0.88 HDAC3 (0.44) HDAC3HDAC1HDAC6F10
SCHEMBL979080 0.88 LMNA (0.44) HDAC3HDAC1HDAC6F10
SCHEMBL978397 0.88 NAMPT (0.46) HDAC3HDAC1HDAC6F10
SCHEMBL975007 0.88 F10 (0.58) HDAC3HDAC1HDAC6F10HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197552-B1 NOVEL TETRAHYDROFUSEDPYRIDINES AS HISTONE DEACETYLASE INHIBITORS 4SC AG (DE) 2012-11-21 EP claimed