SCHEMBL13825293

SCHEMBL13825293

Nc1ccc2c(c1OS(=O)(=O)C(F)(F)F)CCN(C(=O)C(F)(F)F)CC2

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.43
ESR2 Q92731 4/20 0.43
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
PKM P14618 1/20 0.35
ABHD6 Q9BV23 7/20 0.33
ADORA1 P30542 1/20 0.32
DRD2 P14416 4/20 0.32
DRD3 P35462 3/20 0.32
ACKR3 P25106 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL506152 0.87 ESR1 (0.44) ESR1ESR2CA12CA1CA2
SCHEMBL506888 0.86 ESR1 (0.43) ESR1ESR2CA12CA1CA2
SCHEMBL506487 0.86 ESR1 (0.43) ESR1ESR2CA12CA1CA2
SCHEMBL10227565 0.86 ESR1 (0.46) ESR1ESR2CA12CA1CA2
SCHEMBL506132 0.86 ESR1 (0.46) ESR1ESR2CA12CA1CA2
SCHEMBL507158 0.84 ESR1 (0.44) ESR1ESR2PKMABHD6ADORA1
SCHEMBL10227563 0.84 ESR1 (0.44) ESR1ESR2CA12CA1CA2
SCHEMBL506389 0.84 ESR1 (0.42) ESR1ESR2CA12CA1CA2
SCHEMBL506848 0.81 ESR1 (0.42) ESR1ESR2PKMABHD6DRD2
SCHEMBL506173 0.79 DRD2 (0.45) ESR1ESR2ABHD6DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924561-B1 6-ARYLALKYLAMINO- 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS LILLY CO ELI (US) 2012-11-14 EP disclosed