SCHEMBL13825396

SCHEMBL13825396

NC1=NC(c2cccc(-c3cccnc3F)c2)(c2ccc(OC(F)F)cc2F)CC1

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.60
CTSD P07339 14/20 0.60
BACE2 Q9Y5Z0 11/20 0.51
KCNH2 Q12809 1/20 0.40
REN P00797 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13825326 0.89 BACE1 (0.72) BACE1CTSDBACE2KCNH2REN
SCHEMBL7863670 0.85 BACE1 (0.80) BACE1CTSDBACE2KCNH2
SCHEMBL13825347 0.82 BACE1 (0.41) BACE1CTSDBACE2KCNH2REN
SCHEMBL13825358 0.81 BACE1 (0.49) BACE1CTSDBACE2KCNH2
Formic Acid SCHEMBL2285459 0.81 BACE1 (0.73) BACE1CTSDBACE2KCNH2
SCHEMBL13825330 0.80 BACE1 (0.46) BACE1CTSDBACE2KCNH2
SCHEMBL13825504 0.78 BACE1 (0.58) BACE1CTSDBACE2KCNH2REN
SCHEMBL2285462 0.76 BACE1 (0.57) BACE1CTSDBACE2REN
SCHEMBL13825389 0.76 BACE1 (0.52) BACE1CTSDBACE2KCNH2REN
SCHEMBL2287204 0.75 BACE1 (1.00) BACE1CTSDBACE2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245019-B1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-11-14 EP disclosed