SCHEMBL1383989

SCHEMBL1383989

CN(C)CC1CC(OCc2ccc(F)cc2)CCC1(O)c1ccccc1O

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.43
OPRM1 P35372 3/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
OPRL1 P41146 2/20 0.39
SLC18A3 Q16572 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27372207 0.92 OPRM1 (0.47) OPRM1OPRD1OPRK1OPRL1
SCHEMBL4663612 0.91 HDAC4 (0.44) HDAC4OPRM1OPRL1SLC18A3
SCHEMBL19517969 0.90 HDAC4 (0.41) HDAC4OPRM1OPRL1SLC18A3
SCHEMBL4663547 0.90 HDAC4 (0.41) HDAC4OPRM1OPRL1SLC18A3
SCHEMBL4663735 0.90 HDAC4 (0.41) HDAC4OPRM1OPRL1SLC18A3
SCHEMBL4663726 0.88 HDAC4 (0.40) HDAC4OPRM1OPRL1SLC18A3
SCHEMBL4664190 0.88 OPRM1 (0.48) OPRM1OPRD1OPRK1OPRL1SLC18A3
SCHEMBL4664126 0.86 OPRM1 (0.42) HDAC4OPRM1OPRD1OPRK1OPRL1
SCHEMBL4664192 0.85 HDAC4 (0.46) HDAC4OPRM1OPRD1OPRK1OPRL1
SCHEMBL4665456 0.85 OPRM1 (0.48) OPRM1OPRD1OPRK1OPRL1SLC18A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4737583-B2 2011-08-03 JP claimed
JP-2004527491-A 2004-09-09 JP claimed
EP-1390023-A2 PHARMACEUTICAL SALTS Grünenthal GmbH (DE) 2004-02-25 EP claimed
WO-2002067651-A2 PHARMACEUTICAL SALTS Grünenthal GmbH (DE) 2002-09-06 WO claimed
WO-2002067916-A2 PHARMACEUTICAL SALTS Grünenthal GmbH (DE) 2002-09-06 WO claimed
EP-1390023-A2 PHARMACEUTICAL SALTS Grünenthal GmbH (DE) 2004-02-25 EP disclosed
WO-2002067651-A2 PHARMACEUTICAL SALTS Grünenthal GmbH (DE) 2002-09-06 WO disclosed
WO-2002067916-A2 PHARMACEUTICAL SALTS Grünenthal GmbH (DE) 2002-09-06 WO disclosed