SCHEMBL13843441

SCHEMBL13843441

N#Cc1c(-c2c(F)cccc2F)n(CCNCl)c2c(=O)[nH]cnc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.38
HTT P42858 1/20 0.38
BRD4 O60885 1/20 0.32
AURKA O14965 1/20 0.30
DAPK3 O43293 1/20 0.30
JAK2 O60674 1/20 0.30
PRKD3 O94806 1/20 0.30
MAP4K4 O95819 1/20 0.30
PAK4 O96013 1/20 0.30
ABL1 P00519 1/20 0.30
CSF1R P07333 1/20 0.30
RET P07949 1/20 0.30
IGF1R P08069 1/20 0.30
MET P08581 1/20 0.30
PDGFRB P09619 1/20 0.30
PIM1 P11309 1/20 0.30
FGFR1 P11362 1/20 0.30
PDGFRA P16234 1/20 0.30
PRKACA P17612 1/20 0.30
FLT1 P17948 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3937645 0.87 PARP1 (0.40) PARP1HTTBRD4LRRK2
SCHEMBL3939618 0.85 HTT (0.34) PARP1HTT
SCHEMBL13843413 0.80 HTT (0.44) PARP1HTTBRD4DAPK3PRKD3
SCHEMBL27616373 0.77 HTT (0.34) PARP1HTT
SCHEMBL3946110 0.75 LRRK2 (0.31) PARP1HTTLRRK2
SCHEMBL3944568 0.75 KDM4E (0.32)
SCHEMBL3946210 0.72 HTT (0.41) HTTBRD4PIM1LRRK2CLK4
Hydrochloric Acid SCHEMBL3937247 0.72 HTT (0.41) HTTBRD4PIM1LRRK2CLK4
SCHEMBL3943935 0.71 KDM4E (0.36) HTTPIM1CLK4
SCHEMBL3937914 0.71 ALDH1A1 (0.50) HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7528140-B2 Substituted pyrrolo[3,2-d]pyrimidines as glycogen synthase kinase (GSK) inhibitors TEIJIN LIMITED (JP) 2009-05-05 US disclosed