SCHEMBL13845573

SCHEMBL13845573

Cn1nc(C(F)(F)F)c(-c2ccc(F)cc2)c1NC(=O)Nc1ccc(F)cc1F

nearest known ligand 0.88

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.88
NPSR1 Q6W5P4 6/20 0.88
MAPK1 P28482 1/20 0.61
KDM4E B2RXH2 4/20 0.58
LMNA P02545 4/20 0.56
HTT P42858 1/20 0.54
GAA P10253 3/20 0.53
CYP1A2 P05177 2/20 0.52
CYP3A4 P08684 2/20 0.52
CYP2D6 P10635 2/20 0.52
CYP2C9 P11712 2/20 0.52
CYP2C19 P33261 2/20 0.52
HPGD P15428 1/20 0.52
GLA P06280 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15107850 0.94 MAPT (1.00) MAPTNPSR1MAPK1KDM4ELMNA
SCHEMBL12417294 0.93 MAPT (0.76) MAPTNPSR1MAPK1KDM4ELMNA
SCHEMBL12508077 0.92 MAPT (0.79) MAPTNPSR1MAPK1KDM4ELMNA
SCHEMBL12417293 0.87 MAPT (0.87) MAPTNPSR1MAPK1KDM4ELMNA
SCHEMBL12417291 0.85 MAPT (0.69) MAPTNPSR1MAPK1KDM4ELMNA
SCHEMBL15107847 0.82 MAPT (0.89) MAPTNPSR1MAPK1KDM4ELMNA
SCHEMBL13845572 0.81 MAPT (0.79) MAPTNPSR1MAPK1KDM4ELMNA
SCHEMBL12507765 0.76 MAPT (1.00) MAPTNPSR1MAPK1KDM4ELMNA
SCHEMBL12417295 0.75 MAPT (0.76) MAPTNPSR1MAPK1KDM4ELMNA
SCHEMBL12417297 0.74 MAPT (0.89) MAPTNPSR1MAPK1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8486987-B2 Mechanism-based small-molecule parasite inhibitors UNIVERSITY OF MEDICINE AND DENTISTRY OF NEW JERSEY (US) 2013-07-16 US disclosed
WO-2009065096-A1 MECHANISM-BASED SMALL-MOLECULE PARASITE INHIBITORS UNIVERSITY OF MEDICINE AND DENTISTRY OF NEW JERSEY (US) 2009-05-22 WO disclosed