SCHEMBL13845987

SCHEMBL13845987

COc1cc(C(=O)N[C@H]2CCCN(C)C2)ccc1N

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 3/20 0.53
CHRNB2 P17787 4/20 0.51
CHRNA4 P43681 4/20 0.51
HDAC4 P56524 2/20 0.48
HDAC6 Q9UBN7 2/20 0.48
MCHR1 Q99705 1/20 0.47
CHRNB4 P30926 2/20 0.47
CHRNA3 P32297 2/20 0.47
DRD4 P21917 2/20 0.47
USP30 Q70CQ3 1/20 0.47
SLC6A2 P23975 1/20 0.47
KCNH2 Q12809 1/20 0.47
DRD2 P14416 1/20 0.47
DRD3 P35462 1/20 0.47
CHRM4 P08173 1/20 0.47
CHRM5 P08912 1/20 0.47
ADRA2C P18825 1/20 0.47
CHRM3 P20309 1/20 0.47
HTR1D P28221 1/20 0.47
ADRA1B P35368 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13846093 1.00 HTR4 (0.53) HTR4CHRNB2CHRNA4HDAC4HDAC6
SCHEMBL3544670 0.94 HTR4 (0.54) HTR4MCHR1USP30CHRM4CHRM5
SCHEMBL13846090 0.94 HTR4 (0.54) HTR4MCHR1USP30CHRM4CHRM5
SCHEMBL13175736 0.94 HTR4 (0.54) HTR4MCHR1USP30CHRM4CHRM5
SCHEMBL13880647 0.91 AURKA (0.52) HTR4MCHR1PTK2
SCHEMBL13175766 0.89 HTR4 (0.50) HTR4USP30CHRM4CHRM5ADRA2C
SCHEMBL28477021 0.89 HDAC4 (0.46) HTR4CHRNB2CHRNA4HDAC4HDAC6
SCHEMBL738237 0.87 HTR4 (0.53) HTR4MCHR1PTK2
SCHEMBL12825174 0.85 KMT2A (0.57)
SCHEMBL1927002 0.85 KMT2A (0.54) HTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009067547-A1 POLO-LIKE KINASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-05-28 WO disclosed