SCHEMBL13845994

SCHEMBL13845994

COCCC/C=C/c1cccc(I)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
APP P05067 5/20 0.50
BACE1 P56817 2/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C19 P33261 2/20 0.39
HPGD P15428 1/20 0.39
CACNA1B Q00975 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
IDO1 P14902 2/20 0.34
CYP2D6 P10635 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP4F2 P78329 1/20 0.33
CYP4A11 Q02928 1/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13845988 0.95 APP (0.49) APPBACE1MEN1KMT2ACYP1A2
SCHEMBL13846023 0.94 APP (0.48) APPBACE1MEN1KMT2ACYP1A2
SCHEMBL7998452 0.83 RELA (0.49) BACE1MEN1KMT2ACYP1A2CYP2C19
SCHEMBL15051289 0.82 APP (0.46) APPIDO1
SCHEMBL15051287 0.82 APP (0.46) APPIDO1
SCHEMBL13846004 0.80 APP (0.46) APPCYP1A2CYP2C19HPGDCACNA1B
SCHEMBL7990042 0.78 RELA (0.47) BACE1MEN1KMT2ACYP1A2CYP2C19
SCHEMBL8000066 0.77 RELA (0.46) BACE1MEN1KMT2ACYP1A2CYP2C19
SCHEMBL13845999 0.77 APP (0.46) APPMEN1KMT2ACACNA1BCHRM2
SCHEMBL15050808 0.74 APP (0.52) APPCACNA1BCHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009064955-A1 MACROCYCLIC TETRAZOLYL HEPATITIS C SERINE PROTEASE INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2009-05-22 WO disclosed