SCHEMBL13849033

SCHEMBL13849033

O=C(NCc1ccccc1)c1cc(Cl)c2ccccc2c1O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.68
HPGD P15428 4/20 0.62
KDM4E B2RXH2 3/20 0.62
KMT2A Q03164 3/20 0.62
MEN1 O00255 1/20 0.62
ALDH1A1 P00352 1/20 0.62
MAPT P10636 1/20 0.62
PKM P14618 1/20 0.62
HTT P42858 1/20 0.62
HSD17B10 Q99714 1/20 0.62
CA12 O43570 2/20 0.53
CA1 P00915 2/20 0.53
CA2 P00918 2/20 0.53
CA9 Q16790 2/20 0.53
CA3 P07451 1/20 0.53
CA4 P22748 1/20 0.53
CA6 P23280 1/20 0.53
CA5A P35218 1/20 0.53
CA7 P43166 1/20 0.53
CA13 Q8N1Q1 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4066967 0.83 EGLN1 (0.66) HSP90AA1KDM4EKMT2AMEN1ALDH1A1
SCHEMBL20677832 0.81 HSP90AA1 (1.00) HSP90AA1HPGDKMT2ACA12CA1
SCHEMBL13656899 0.79 MEN1 (0.66) HPGDKDM4EKMT2AMEN1ALDH1A1
SCHEMBL5860823 0.78 NPC1 (0.71) HSP90AA1HPGDKMT2AALDH1A1LMNA
SCHEMBL485443 0.77 HSD17B10 (1.00) HPGDKDM4EKMT2AMEN1ALDH1A1
SCHEMBL9400432 0.77 EGLN1 (0.66) HPGDKDM4EKMT2AMEN1MAPT
SCHEMBL11316839 0.77 NAAA (0.59) HPGDKDM4EKMT2AMEN1ALDH1A1
SCHEMBL11598238 0.77 NAAA (0.59) HPGDKDM4EKMT2AMEN1ALDH1A1
SCHEMBL9095008 0.77 HPGD (0.51) HSP90AA1HPGDKDM4EKMT2AMEN1
SCHEMBL9095674 0.76 KDM4E (0.52) HSP90AA1HPGDKDM4EKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1326865-B1 AZA- AND POLYAZA-NAPHTHALENYL CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2009-05-06 EP disclosed