SCHEMBL13858261

SCHEMBL13858261

Nc1ccnc(C2CCNCC2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.49
MKNK1 Q9BUB5 3/20 0.48
MKNK2 Q9HBH9 3/20 0.48
CCNT1 O60563 2/20 0.44
CDK9 P50750 2/20 0.44
ROCK1 Q13464 2/20 0.41
TLR9 Q9NR96 3/20 0.41
TLR8 Q9NR97 3/20 0.41
TLR7 Q9NYK1 3/20 0.41
HRH3 Q9Y5N1 1/20 0.41
ROCK2 O75116 1/20 0.38
ASIC3 Q9UHC3 1/20 0.38
ADORA2A P29274 2/20 0.38
ADORA1 P30542 2/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
PKM P14618 1/20 0.38
ALOX15 P16050 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31302450 0.90 MKNK1 (0.43) HRH4MKNK1MKNK2CCNT1CDK9
SCHEMBL12068738 0.87 ADORA2A (0.45) MKNK1MKNK2ASIC3ADORA2AADORA1
SCHEMBL4183278 0.83 CHRNA7 (0.42) HRH4HRH3ASIC3ADORA2AADORA1
SCHEMBL29851723 0.83 CHRNA7 (0.46) HRH4ASIC3ADORA2AADORA1ALDH1A1
SCHEMBL18957072 0.83 CHRNA7 (0.46) HRH4ASIC3ADORA2AADORA1ALDH1A1
SCHEMBL30073115 0.81 KDM4E (0.44) HRH4ASIC3ADORA2AADORA1ALDH1A1
SCHEMBL18956812 0.81 KDM4E (0.44) HRH4ASIC3ADORA2AADORA1ALDH1A1
SCHEMBL23612242 0.80 CHEK1 (0.52) ROCK1ROCK2MAP3K12
SCHEMBL29988658 0.80 CHEK1 (0.52) ROCK1ROCK2MAP3K12
SCHEMBL3388660 0.79 ASIC3 (0.44) MKNK1MKNK2ASIC3ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012158784-A2 MODULATORS OF THE NUCLEAR HORMONE RECEPTOR ROR KAMENECKA THEODORE MARK (US) 2012-11-22 WO disclosed