SCHEMBL13862004

SCHEMBL13862004

CC(C)c1ccc(C(=O)Nc2cn3cc(-c4cnco4)ccc3n2)cn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK2 P49760 6/20 0.52
CLK1 P49759 4/20 0.52
MAP3K5 Q99683 9/20 0.46
MCHR1 Q99705 1/20 0.44
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 1/20 0.43
PKM P14618 1/20 0.43
DYRK1A Q13627 3/20 0.43
HRH1 P35367 2/20 0.43
WNT1 P04628 1/20 0.43
GSK3B P49841 1/20 0.43
PDGFRB P09619 1/20 0.43
KIT P10721 1/20 0.43
PDGFRA P16234 1/20 0.43
FLT3 P36888 1/20 0.43
CLK3 P49761 1/20 0.43
SIK2 Q9H0K1 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
DYRK1B Q9Y463 1/20 0.43
HTR1A P08908 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3486095 0.85 CLK2 (0.73) CLK2CLK1MAP3K5MCHR1DYRK1A
Hydrochloric Acid SCHEMBL3486014 0.84 CLK2 (0.72) CLK2CLK1MAP3K5DYRK1AHRH1
SCHEMBL3486108 0.82 MAP3K5 (0.67) CLK2CLK1MAP3K5DYRK1AHRH1
Hydrochloric Acid SCHEMBL3485471 0.82 MAP3K5 (0.66) CLK2CLK1MAP3K5DYRK1AHRH1
SCHEMBL17632607 0.74 PIK3CA (0.44) CLK2CLK1MAP3K5KDM4ENPC1
SCHEMBL3779466 0.68 CYP2C9 (0.61) KDM4ENPC1PKM
SCHEMBL19296078 0.67 LMNA (0.56) MCHR1KDM4ENPC1PKM
SCHEMBL3485541 0.67 CLK2 (0.80) CLK2CLK1MAP3K5DYRK1AHRH1
SCHEMBL17632835 0.66 USP30 (0.51) DYRK1AWNT1GSK3B
SCHEMBL17632833 0.66 USP30 (0.51) DYRK1AWNT1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058309-A1 FUSED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-05-13 EP disclosed