SCHEMBL13862010

SCHEMBL13862010

CC(C)(C)C1C=CC(C(=O)Nc2cn3nc(-c4ccc5c(c4)OCO5)ccc3n2)=CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 6/20 0.40
ADORA1 P30542 5/20 0.40
PIK3CG P48736 4/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 3/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
KMT2A Q03164 2/20 0.39
FYN P06241 2/20 0.39
ADORA2A P29274 2/20 0.38
LMNA P02545 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CSNK1D P48730 2/20 0.38
CSNK1E P49674 2/20 0.38
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13498819 0.80 MAP3K5 (0.52) ADORA3ADORA1POLBMAPTNPC1
Formic Acid SCHEMBL3485941 0.77 MAP3K5 (0.48) ADORA3ADORA1POLBMAPTNPC1
SCHEMBL3091747 0.63 PIK3CG (0.63) ADORA3ADORA1PIK3CG
SCHEMBL13498813 0.62 MAP3K5 (0.56) ADORA3MAPTCSNK1DCSNK1E
SCHEMBL3485946 0.62 ALDH1A1 (0.46) ADORA3ADORA1POLBMAPTNPC1
SCHEMBL3486280 0.61 MAP3K5 (0.67) POLBMAPTLMNACSNK1DCSNK1E
SCHEMBL13498806 0.60 MAP3K5 (0.57) CSNK1DCSNK1E
SCHEMBL13498805 0.60 MAP3K5 (0.56) CSNK1DCSNK1ERIPK1
SCHEMBL3487219 0.60 CSNK1D (0.56) CSNK1DCSNK1E
SCHEMBL12664264 0.59 CSNK1D (0.52) CSNK1DCSNK1ERIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058309-A1 FUSED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-05-13 EP disclosed