SCHEMBL13864488

SCHEMBL13864488

C=Cc1cccc(-c2nc3ccccc3nc2O[C@@H]2C[C@@H](C(=O)OC)N(C(=O)[C@@H](NC(=O)OCC(F)(F)C=C)C(C)(C)C)C2)c1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.34
ELANE P08246 2/20 0.33
KIF11 P52732 1/20 0.32
KCNH2 Q12809 1/20 0.32
DHODH Q02127 2/20 0.31
CTSB P07858 1/20 0.31
PPP3CB P16298 1/20 0.31
BIRC2 Q13490 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13864551 0.94 CYP3A4 (0.35) CYP3A4ELANECTSBPPP3CBBIRC2
SCHEMBL13864478 0.90 CYP3A4 (0.36) CYP3A4ELANEKIF11KCNH2DHODH
SCHEMBL7999134 0.89 CYP3A4 (0.42) CYP3A4ELANE
SCHEMBL13864540 0.89 CYP3A4 (0.35) CYP3A4ELANEKIF11KCNH2DHODH
SCHEMBL10261387 0.87 CYP3A4 (0.34) CYP3A4ELANEBIRC2
SCHEMBL10261079 0.87 CYP3A4 (0.34) CYP3A4ELANEBIRC2
SCHEMBL8014416 0.83 CYP3A4 (0.33) CYP3A4ELANE
SCHEMBL8010213 0.83 CYP3A4 (0.33) CYP3A4ELANE
SCHEMBL8008173 0.83 MMP2 (0.32) CYP3A4
SCHEMBL13864577 0.82 ELANE (0.32) CYP3A4ELANEKIF11KCNH2CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8951998-B2 Quinoxaline-containing compounds as hepatitis C virus inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2015-02-10 US disclosed
US-8951998-B2 Quinoxaline-containing compounds as hepatitis C virus inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2015-02-10 US disclosed
US-8324155-B2 Quinoxaline-containing compounds as hepatitis C virus inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2012-12-04 US disclosed
WO-2009064975-A1 QUINOXALINE-CONTAINING COMPOUNDS AS HEPATITIS C VIRUS INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2009-05-22 WO disclosed