SCHEMBL13865181

SCHEMBL13865181

Bc1oc(-c2nn(Cc3ccccc3F)c3ccccc23)nc1C(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BUB1 O43683 15/20 0.44
CHRM1 P11229 2/20 0.41
GUCY1A1 Q02108 3/20 0.39
GUCY1B1 Q02153 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13865218 0.79 BUB1 (0.48) BUB1CHRM1
SCHEMBL13865195 0.79 BUB1 (0.46) BUB1CHRM1GUCY1A1GUCY1B1
SCHEMBL4425532 0.76 BUB1 (0.45) BUB1CHRM1
SCHEMBL13865194 0.76 BUB1 (0.45) BUB1CHRM1
SCHEMBL13865208 0.75 BUB1 (0.48) BUB1CHRM1
SCHEMBL13865183 0.75 CYP2D6 (0.52) BUB1CHRM1
SCHEMBL4434101 0.74 BUB1 (0.45) BUB1CHRM1
SCHEMBL4426683 0.74 BUB1 (0.43) BUB1CHRM1
SCHEMBL13865201 0.74 BUB1 (0.45) BUB1CHRM1
SCHEMBL13865192 0.73 BUB1 (0.46) BUB1CHRM1GUCY1A1GUCY1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934311-B1 NEW HETEROCYCLYLMETHYL-SUBSTITUTED PYRAZOL DERIVATES BAYER HEALTHCARE AG (DE) 2009-05-13 EP disclosed