SCHEMBL13865191

SCHEMBL13865191

Fc1ccccc1Cn1nc(-c2nc(-c3ccccc3)co2)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
BUB1 O43683 13/20 0.46
CHRM1 P11229 2/20 0.45
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
SCN8A Q9UQD0 1/20 0.42
TP53 P04637 1/20 0.41
GAA P10253 1/20 0.41
GUCY1A1 Q02108 2/20 0.40
GUCY1B1 Q02153 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13865211 0.85 CYP2D6 (0.57) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL13865208 0.84 BUB1 (0.48) BUB1CHRM1CYP1A2CYP2D6
SCHEMBL13865193 0.83 BUB1 (0.45) BUB1CHRM1CYP1A2CYP3A4CYP2D6
SCHEMBL13865226 0.83 BUB1 (0.51) KMT2ABUB1CHRM1GUCY1A1GUCY1B1
SCHEMBL13865192 0.82 BUB1 (0.46) MEN1KMT2ABUB1CHRM1GUCY1A1
SCHEMBL13865196 0.81 BUB1 (0.46) BUB1CHRM1
SCHEMBL13865195 0.81 BUB1 (0.46) BUB1CHRM1GUCY1A1GUCY1B1
SCHEMBL13865223 0.81 BUB1 (0.43) BUB1CHRM1CYP1A2CYP3A4CYP2D6
SCHEMBL13865217 0.80 BUB1 (0.43) BUB1CHRM1CYP1A2CYP3A4CYP2D6
SCHEMBL13865212 0.79 BUB1 (0.43) BUB1CHRM1CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934311-B1 NEW HETEROCYCLYLMETHYL-SUBSTITUTED PYRAZOL DERIVATES BAYER HEALTHCARE AG (DE) 2009-05-13 EP disclosed