SCHEMBL13865205

SCHEMBL13865205

Fc1ccccc1Cn1nc(-c2nnc(CCl)o2)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 2/20 0.46
BUB1 O43683 13/20 0.45
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
SCN8A Q9UQD0 1/20 0.40
PDE5A O76074 2/20 0.40
GRM2 Q14416 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13865189 0.89 BUB1 (0.45) CHRM1BUB1ALDH1A1LMNACYP1A2
SCHEMBL13865188 0.84 PDE5A (0.55) CHRM1ALDH1A1LMNACYP1A2CYP3A4
SCHEMBL13865218 0.76 BUB1 (0.48) CHRM1BUB1ALDH1A1CYP1A2CYP3A4
SCHEMBL13865192 0.74 BUB1 (0.46) CHRM1BUB1
SCHEMBL5565576 0.74 PDE5A (0.61) ALDH1A1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL13865208 0.74 BUB1 (0.48) CHRM1BUB1ALDH1A1CYP1A2CYP2D6
SCHEMBL13865183 0.74 CYP2D6 (0.52) CHRM1BUB1ALDH1A1CYP1A2CYP3A4
SCHEMBL13865194 0.73 BUB1 (0.45) CHRM1BUB1ALDH1A1LMNACYP1A2
SCHEMBL4425532 0.73 BUB1 (0.45) CHRM1BUB1ALDH1A1LMNACYP1A2
SCHEMBL13865191 0.72 MEN1 (0.46) CHRM1BUB1CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934311-B1 NEW HETEROCYCLYLMETHYL-SUBSTITUTED PYRAZOL DERIVATES BAYER HEALTHCARE AG (DE) 2009-05-13 EP disclosed