SCHEMBL13865458

SCHEMBL13865458

Brc1ccc(C(c2ccccc2)c2ccc(Br)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.60
ALDH1A1 P00352 3/20 0.53
TDP1 Q9NUW8 1/20 0.53
SLC6A2 P23975 4/20 0.50
SLC6A4 P31645 4/20 0.50
SLC6A3 Q01959 4/20 0.50
MAPK1 P28482 1/20 0.50
HDAC1 Q13547 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
CFTR P13569 1/20 0.44
GOPC Q9HD26 1/20 0.44
CYP2A6 P11509 1/20 0.44
OPRM1 P35372 2/20 0.44
CHRM2 P08172 1/20 0.44
HTR1A P08908 1/20 0.44
ADRA2A P08913 1/20 0.44
CHRM1 P11229 1/20 0.44
DRD1 P21728 1/20 0.44
TBXA2R P21731 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3692372 1.00 HTR2A (0.60) HTR2AALDH1A1TDP1SLC6A2SLC6A4
SCHEMBL1989430 0.88 CYP2A6 (0.57) HTR2AALDH1A1TDP1MAPK1CYP2A6
SCHEMBL19669010 0.87 ALDH1A1 (0.71) HTR2AALDH1A1TDP1SLC6A2SLC6A4
SCHEMBL16229373 0.87 ALDH1A1 (0.71) HTR2AALDH1A1TDP1SLC6A2SLC6A4
SCHEMBL2956444 0.85 SLC6A2 (0.63) HTR2ASLC6A2SLC6A4SLC6A3HDAC1
SCHEMBL13721485 0.85 HTR2A (0.47) HTR2AALDH1A1TDP1SLC6A2SLC6A4
SCHEMBL18481572 0.83 CYP2A6 (0.54) HTR2ASLC6A2SLC6A4SLC6A3CYP2A6
SCHEMBL144 0.82 SLC6A2 (0.67) HTR2ASLC6A2SLC6A4SLC6A3MAPK1
SCHEMBL11576225 0.81 HTR2A (0.58) HTR2AALDH1A1TDP1SLC6A2SLC6A4
SCHEMBL24238343 0.79 HTR2A (0.61) HTR2AALDH1A1TDP1SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7531573-B2 potent, selective and safe inhibitors of the Ca2+-activated potassium channel CHILDREN'S MEDICAL CENTER CORPORATION (US) 2009-05-12 US disclosed
US-7531573-B2 potent, selective and safe inhibitors of the Ca2+-activated potassium channel CHILDREN'S MEDICAL CENTER CORPORATION (US) 2009-05-12 US disclosed