SCHEMBL13868378

SCHEMBL13868378

CCC1CN(Cc2ccccc2)C(=O)CN1C(C)=O

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 14/20 0.60
BRS3 P32247 1/20 0.48
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.45
TSHR P16473 1/20 0.45
ABCB1 P08183 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13868377 0.90 BRD4 (0.50) BRD4BRS3ALDH1A1HPGDTSHR
SCHEMBL13868376 0.83 BRS3 (0.52) BRD4BRS3ALDH1A1HPGDTSHR
SCHEMBL3906448 0.79 HTT (0.46) BRD4BRS3
SCHEMBL21224119 0.78 CACNA1G (0.56) BRD4ALDH1A1HPGDTSHR
SCHEMBL21224116 0.78 CACNA1G (0.56) BRD4ALDH1A1HPGDTSHR
SCHEMBL13868382 0.73 BRD4 (0.45) BRD4BRS3ALDH1A1HPGDABCB1
SCHEMBL8572660 0.73 KLK7 (0.40) BRD4ALDH1A1HPGDTSHR
SCHEMBL8572656 0.73 KLK7 (0.40) BRD4ALDH1A1HPGDTSHR
SCHEMBL3914346 0.72 HTT (0.54) BRD4ALDH1A1
SCHEMBL22536521 0.71 CACNA1G (0.49) BRD4ALDH1A1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7517532-B2 Dihydroxypyridopyrazine-1,6-dione compounds useful as HIV integrase inhibitors MERCK & CO., INC. (US) 2009-04-14 US disclosed