SCHEMBL1386959

SCHEMBL1386959

Cc1c(S(=O)(=O)Nc2ccc(Cl)cc2)c2cc(C#N)ccc2n1CC(=O)O

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 17/20 0.54
AKR1B1 P15121 5/20 0.54
CYP2C9 P11712 1/20 0.43
ALDH1A1 P00352 1/20 0.42
MAPK1 P28482 1/20 0.42
STAT3 P40763 1/20 0.42
PTGES O14684 1/20 0.42
ALOX5 P09917 1/20 0.42
FLT1 P17948 1/20 0.41
FLT4 P35916 1/20 0.41
KDR P35968 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6533614 0.87 PTGDR2 (0.71) PTGDR2AKR1B1CYP2C9
SCHEMBL5476456 0.85 PTGDR2 (0.72) PTGDR2AKR1B1
SCHEMBL1384482 0.85 PTGDR2 (0.75) PTGDR2AKR1B1CYP2C9ALDH1A1MAPK1
SCHEMBL5477529 0.78 PTGDR2 (0.62) PTGDR2AKR1B1CYP2C9
SCHEMBL5438307 0.76 PTGDR2 (0.60) PTGDR2AKR1B1CYP2C9
SCHEMBL1406046 0.76 PTGDR2 (0.78) PTGDR2AKR1B1CYP2C9
SCHEMBL5428186 0.75 PTGDR2 (0.61) PTGDR2CYP2C9
SCHEMBL5474079 0.74 PTGDR2 (0.63) PTGDR2AKR1B1CYP2C9
SCHEMBL3010082 0.74 PTGDR2 (0.46) PTGDR2AKR1B1CYP2C9ALDH1A1MAPK1
SCHEMBL5474051 0.74 PTGDR2 (0.56) PTGDR2AKR1B1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4791729-B2 2011-10-12 JP claimed
JP-2005537265-A 2005-12-08 JP claimed
EP-1551802-A1 INDOLE-3-SULPHUR DERIVATIVES AstraZeneca AB (SE) 2005-07-13 EP claimed
WO-2004007451-A1 INDOLE-3-SULPHUR DERIVATIVES ASTRAZENECA AB (SE) 2004-01-22 WO claimed