SCHEMBL13873266

SCHEMBL13873266

COC(=O)c1ccc(C(=O)OC)c(Nc2nc(Nc3ccc(NC(C)=O)cc3)ncc2N=O)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.49
ALDH1A1 P00352 4/20 0.49
HPGD P15428 2/20 0.49
CASP1 P29466 1/20 0.49
CASP7 P55210 1/20 0.49
HSD17B10 Q99714 1/20 0.49
CYP2C9 P11712 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C19 P33261 1/20 0.44
MCL1 Q07820 1/20 0.44
PTK2B Q14289 1/20 0.44
PTK2 Q05397 1/20 0.43
AURKA O14965 3/20 0.43
PLK1 P53350 1/20 0.43
HDAC1 Q13547 1/20 0.43
SYK P43405 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4023425 0.83 MAPT (0.68) KDM4EALDH1A1HPGDCASP1CASP7
Hydrochloric Acid SCHEMBL3814476 0.83 MAPT (0.67) KDM4EALDH1A1HPGDCASP1CASP7
SCHEMBL13809932 0.77 PLK1 (0.70) CYP2C9MEN1KMT2ACYP1A2CYP3A4
SCHEMBL13872996 0.76 PLK1 (0.51) KDM4EALDH1A1HPGDCYP2C9MEN1
SCHEMBL13873249 0.76 PLK1 (0.56) MEN1KMT2APTK2BPTK2PLK1
SCHEMBL13873254 0.72 PTK2 (0.68) PTK2BPTK2AURKAPLK1SYK
SCHEMBL4031609 0.70 MAPT (0.70) CYP2C9MEN1KMT2ACYP1A2CYP3A4
Hydrochloric Acid SCHEMBL3814985 0.69 MAPT (0.69) CYP2C9MEN1KMT2ACYP1A2CYP3A4
SCHEMBL13088436 0.69 KDM4E (0.69) KDM4EALDH1A1HPGDCASP1CASP7
SCHEMBL30487008 0.69 KDM4E (0.69) KDM4EALDH1A1HPGDCASP1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7514446-B2 Pyrimidine compounds SMITHKLINE BEECHAM CORPORATION (US) 2009-04-07 US disclosed