SCHEMBL13874403

SCHEMBL13874403

CNc1cccc(N2CCN(c3ncnc4ccc(-c5cn[nH]c5)cc34)CC2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 16/20 0.49
CYP3A4 P08684 16/20 0.49
CLK4 Q9HAZ1 13/20 0.49
ALDH1A1 P00352 10/20 0.49
LMNA P02545 8/20 0.49
HIF1A Q16665 8/20 0.49
MAPK1 P28482 7/20 0.49
MEN1 O00255 7/20 0.49
KMT2A Q03164 7/20 0.49
AKT1 P31749 1/20 0.49
USP2 O75604 9/20 0.48
CYP2C19 P33261 7/20 0.48
CYP2D6 P10635 6/20 0.48
HSD17B10 Q99714 1/20 0.48
ALOX15 P16050 1/20 0.47
TSHR P16473 3/20 0.46
KDM4E B2RXH2 3/20 0.45
HPGD P15428 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
RPS6KB1 P23443 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4714577 0.87 CYP1A2 (0.51) CYP1A2CYP3A4CLK4ALDH1A1LMNA
Hydrochloric Acid SCHEMBL3849363 0.86 CYP1A2 (0.50) CYP1A2CYP3A4CLK4ALDH1A1LMNA
SCHEMBL5853346 0.86 AKT1 (0.54) CYP1A2CYP3A4CLK4ALDH1A1LMNA
SCHEMBL3855266 0.85 AKT1 (0.59) CYP1A2CYP3A4CLK4ALDH1A1LMNA
Hydrochloric Acid SCHEMBL3851639 0.85 ACHE (0.54) CYP1A2CYP3A4CLK4ALDH1A1LMNA
SCHEMBL3846924 0.83 AKT1 (0.51) CYP1A2CYP3A4CLK4ALDH1A1LMNA
SCHEMBL4716295 0.83 CYP1A2 (0.50) CYP1A2CYP3A4CLK4ALDH1A1LMNA
Trifluoroacetic Acid SCHEMBL3846430 0.83 AKT1 (0.48) CYP1A2CYP3A4CLK4ALDH1A1LMNA
Trifluoroacetic Acid SCHEMBL3855041 0.82 CYP1A2 (0.58) CYP1A2CYP3A4CLK4ALDH1A1LMNA
Hydrochloric Acid SCHEMBL3846099 0.82 AKT1 (0.48) CYP1A2CYP3A4CLK4ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed