SCHEMBL13875673

SCHEMBL13875673

Cn1c(=O)[nH]c2c(N3CCNCC3)nc(O)nc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.40
CHRNB2 P17787 1/20 0.39
ADRA1D P25100 1/20 0.39
HTR1E P28566 1/20 0.39
CHRNA3 P32297 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRK1 P41145 1/20 0.39
POLB P06746 1/20 0.39
SIRT5 Q9NXA8 1/20 0.39
ALDH1A1 P00352 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
CASP1 P29466 1/20 0.34
CYP2C19 P33261 1/20 0.34
CASP7 P55210 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13866874 0.83 DPP4 (0.42) DPP4CHRNB2ADRA1DHTR1ECHRNA3
SCHEMBL13875751 0.83 HRH4 (0.51) DPP4CHRNB2ADRA1DHTR1ECHRNA3
SCHEMBL13875671 0.81 DPP4 (0.38) DPP4CHRNB2ADRA1DHTR1ECHRNA3
SCHEMBL13875841 0.81 DPP4 (0.38) DPP4CHRNB2ADRA1DHTR1ECHRNA3
SCHEMBL13875837 0.81 DPP4 (0.38) DPP4CHRNB2ADRA1DHTR1ECHRNA3
SCHEMBL13875848 0.81 ADRB1 (0.41) DPP4CHRNB2ADRA1DHTR1ECHRNA3
SCHEMBL13875846 0.78 TLR7 (0.41) DPP4CHRNB2ADRA1DHTR1ECHRNA3
SCHEMBL13875749 0.78 DPP4 (0.39) DPP4CHRNB2ADRA1DHTR1ECHRNA3
SCHEMBL13875849 0.78 DPP4 (0.39) DPP4CHRNB2ADRA1DHTR1ECHRNA3
Trifluoroacetic Acid SCHEMBL3877706 0.77 DPP4 (0.39) DPP4CHRNB2ADRA1DHTR1ECHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7524847-B2 Fused 1,3-dihydro-imidazole ring compounds EISAI R&D MANAGEMENT CO., LTD. (JP) 2009-04-28 US disclosed