SCHEMBL1389215

SCHEMBL1389215

O=[C]N1C=Cc2ccccc2C1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.38
HSD17B3 P37058 1/20 0.35
PARP1 P09874 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
RXFP1 Q9HBX9 1/20 0.31
NOTUM Q6P988 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1014977 0.81 CA1 (0.41) HDAC3HSD17B3PARP1CA1CA2
Hydrochloric Acid SCHEMBL7007188 0.79 CA1 (0.40) HDAC3HSD17B3PARP1CA1CA2
SCHEMBL28632594 0.79 CA1 (0.40) HDAC3HSD17B3PARP1CA1CA2
SCHEMBL22777551 0.73 HDAC3 (0.36) HDAC3HSD17B3PARP1CA1CA2
SCHEMBL3069885 0.73 HDAC3 (0.43) HDAC3HSD17B3PARP1CA1CA2
SCHEMBL143063 0.69 HDAC3 (0.38) HDAC3HSD17B3PARP1CA1CA2
SCHEMBL1564351 0.69 HDAC3 (0.41) HDAC3HSD17B3PARP1CA1CA2
SCHEMBL13932579 0.69 HDAC3 (0.38) HDAC3HSD17B3PARP1CA1CA2
SCHEMBL11353696 0.69 HDAC3 (0.38) HDAC3HSD17B3PARP1CA1CA2
SCHEMBL4854749 0.69 HDAC3 (0.41) HDAC3HSD17B3PARP1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3750886-A1 TETRAHYDROISOQUINOLINE COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION CONTAINING SAME, AND USE THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2020-12-16 EP claimed
JP-2011529031-A 2011-12-01 JP claimed
EP-2318355-A1 1,1'-DIADAMANTYL CARBOXYLIC ACIDS, MEDICAMENTS CONTAINING SUCH COMPOUNDS AND THEIR USE Boehringer Ingelheim International GmbH (DE) 2011-05-11 EP claimed
WO-2010010174-A1 1,1'-DIADAMANTYL CARBOXYLIC ACIDS, MEDICAMENTS CONTAINING SUCH COMPOUNDS AND THEIR USE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-01-28 WO claimed
EP-1027351-B1 PHENANTHROLINE DERIVATIVES FIBROGEN INC (US) 2003-12-03 EP claimed
CN-110467629-A Quinone derivatives, its pharmaceutical composition and application SHANGHAI DE NOVO PHARMATECH CO LTD 2019-11-19 CN disclosed
EP-1940838-A1 TRIAZOLOPYRIDINE DERIVATIVES AS INHIBITORS OF LIPASES AND PHOSPHOLIPASES sanofi-aventis (FR) 2008-07-09 EP disclosed
WO-2007045392-A1 TRIAZOLOPYRIDINE DERIVATIVES AS INHIBITORS OF LIPASES AND PHOSPHOLIPASES SANOFI-AVENTIS (DE) 2007-04-26 WO disclosed
WO-2006099610-A2 METHODS OF IDENTIFYING THERAPEUTIC TARGETS FOR THE TREATMENT OF VULVOVAGINAL ATROPHY WYETH (US) 2006-09-21 WO disclosed