SCHEMBL13893967

SCHEMBL13893967

Cc1ccc2c(=O)n(-c3cccc(B4OC(C)(C)C(C)(C)O4)c3C)cnc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 12/20 0.47
JAK2 O60674 3/20 0.47
POLB P06746 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HCAR1 Q9BXC0 2/20 0.35
TP53 P04637 1/20 0.35
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12070562 0.90 BTK (0.50) BTKJAK2POLBHCAR1
SCHEMBL29709475 0.88 BTK (0.52) BTKJAK2POLBMEN1KMT2A
SCHEMBL9983255 0.88 BTK (0.52) BTKJAK2POLBMEN1KMT2A
SCHEMBL708646 0.88 BTK (0.49) BTKJAK2POLBMEN1KMT2A
SCHEMBL149181 0.83 BTK (0.50) BTKJAK2POLBHCAR1
SCHEMBL29709471 0.83 BTK (0.50) BTKJAK2POLBHCAR1
SCHEMBL9983905 0.79 BTK (0.59) BTKJAK2POLBHCAR1
SCHEMBL12070563 0.77 BTK (0.50) BTKJAK2KMT2A
SCHEMBL8737267 0.75 BTK (0.45) BTKJAK2POLBHCAR1
SCHEMBL17645752 0.71 BTK (0.49) BTKJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009053269-A1 NOVEL KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2009-04-30 WO disclosed