SCHEMBL13900421

SCHEMBL13900421

CC(=O)c1cccc(-c2ccccc2NC(=O)CCNC(=O)OC(C)(C)C)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
KMT2A Q03164 5/20 0.43
SUCNR1 Q9BXA5 2/20 0.43
GAA P10253 2/20 0.43
HDAC3 O15379 3/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC2 Q92769 2/20 0.42
HDAC10 Q969S8 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
NCOR2 Q9Y618 1/20 0.42
SOAT1 P35610 2/20 0.41
SELP P16109 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
MALT1 Q9UDY8 1/20 0.40
ALDH1A1 P00352 4/20 0.40
NPSR1 Q6W5P4 2/20 0.40
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 3/20 0.40
MEN1 O00255 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4048733 0.94 CA1 (0.52) CA1CA2SUCNR1HDAC3HDAC1
SCHEMBL16747675 0.82 GAA (0.61) CA1CA2KMT2AGAATDP1
SCHEMBL6831601 0.81 SOAT1 (0.44) CA1CA2KMT2AGAAHDAC3
SCHEMBL4051518 0.80 KCNA5 (0.50) KMT2ASUCNR1MALT1
SCHEMBL4060683 0.78 KCNA5 (0.50) SUCNR1HDAC1HDAC10HDAC6MALT1
SCHEMBL8692644 0.77 POLB (0.55) CA1CA2KMT2AGAATDP1
SCHEMBL13233342 0.76 CA1 (0.49) CA1CA2KMT2AGAAHDAC3
SCHEMBL5583416 0.76 ALDH1A1 (0.56) CA1CA2KMT2AHDAC3HDAC1
SCHEMBL18535719 0.75 BRD9 (0.50) KMT2AALDH1A1NPSR1HTTL3MBTL1
SCHEMBL9524622 0.75 CYP1A2 (0.59) CA1CA2KMT2AALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7507753-B2 melanocortin receptor agonist, antagonist; preventing or treating inflammatory diseases, AIDS, obesity, bulimia, anorexia or sexual dysfunction; N-(2-aminoethyl)-3'-[1-{N-(1-benzylpiperidin-4-yl)-N-(2-naphthylacetyl)aminoethyl][1,1'-biphenyl)-2-carboxamide dihydrochloride TAKEDA CHEMICAL INDUSTRIES LTD. (JP) 2009-03-24 US disclosed