SCHEMBL13902801

SCHEMBL13902801

CCOC(=O)c1cccc(Cc2cc(Cl)ccc2CCc2ccccc2Cl)n1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 14/20 0.54
CYP1A2 P05177 5/20 0.48
CYP2C9 P11712 4/20 0.47
GABRA2 P47869 2/20 0.46
GABRB2 P47870 2/20 0.46
CYP2C19 P33261 2/20 0.44
CYP3A4 P08684 1/20 0.44
TBXA2R P21731 1/20 0.44
PTGS1 P23219 1/20 0.44
PTGER3 P43115 1/20 0.44
PTGER2 P43116 1/20 0.44
MAPT P10636 1/20 0.44
MRGPRX4 Q96LA9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13902798 0.86 PTGER1 (0.50) PTGER1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL2954986 0.85 PTGER1 (0.77) PTGER1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL2955012 0.82 CYP1A2 (0.55) PTGER1CYP1A2CYP2C9CYP2C19CYP3A4
Acetone SCHEMBL27709152 0.80 CYP1A2 (0.52) PTGER1CYP1A2CYP2C9CYP2C19TBXA2R
SCHEMBL3212344 0.80 PTGER1 (0.55) PTGER1CYP1A2CYP2C9CYP2C19TBXA2R
SCHEMBL2960944 0.79 PTGER1 (0.77) PTGER1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL14397613 0.78 CYP1A2 (0.52) PTGER1CYP1A2CYP2C9CYP2C19TBXA2R
SCHEMBL2962415 0.77 PTGER1 (0.58) PTGER1CYP1A2CYP2C9CYP2C19TBXA2R
SCHEMBL2961468 0.77 PTGER1 (0.77) PTGER1CYP1A2CYP2C9CYP2C19TBXA2R
SCHEMBL2949627 0.77 PTGER1 (0.78) PTGER1CYP1A2CYP2C9CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833795-B1 PYRIDINE COMPOUNDS FOR THE TREATMENT OF PROSTAGLANDIN MEDIATED DISEASES GLAXO GROUP LTD (GB) 2009-03-04 EP disclosed