SCHEMBL13909591

SCHEMBL13909591

COc1cccnc1CNCc1ccc(CNC2CCCc3cccnc32)cc1

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.57
HDAC6 Q9UBN7 2/20 0.57
KDM4E B2RXH2 3/20 0.44
CXCR4 P61073 8/20 0.44
ADORA2A P29274 1/20 0.44
DRD2 P14416 1/20 0.40
KMT2A Q03164 1/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13909513 0.89 HDAC1 (0.54) HDAC1HDAC6KDM4ECXCR4ADORA2A
SCHEMBL13909588 0.86 HDAC1 (0.60) HDAC1HDAC6KDM4ECXCR4CYP3A4
SCHEMBL13909590 0.84 HDAC1 (0.62) HDAC1HDAC6KDM4ECXCR4CYP3A4
SCHEMBL14037709 0.84 HDAC1 (0.64) HDAC1HDAC6KDM4ECXCR4ADORA2A
SCHEMBL13909820 0.83 HDAC1 (0.76) HDAC1HDAC6KDM4ECXCR4CYP3A4
SCHEMBL29823139 0.80 HDAC1 (0.62) HDAC1HDAC6KDM4ECXCR4CYP3A4
SCHEMBL1882612 0.80 HDAC1 (0.62) HDAC1HDAC6KDM4ECXCR4CYP3A4
Bromide SCHEMBL4543315 0.79 HDAC1 (0.61) HDAC1HDAC6KDM4ECXCR4CYP3A4
SCHEMBL4887341 0.79 HDAC1 (0.69) HDAC1HDAC6KDM4ECXCR4CYP3A4
SCHEMBL4562865 0.79 HDAC1 (0.69) HDAC1HDAC6KDM4ECXCR4CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317445-B1 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS ANORMED INC (CA) 2009-03-11 EP disclosed