SCHEMBL13915596

SCHEMBL13915596

COc1cc2c(Cl)c(C(N)=O)cnc2cc1OC(=O)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 19/20 0.57
NUDT1 P36639 1/20 0.48
EGFR P00533 1/20 0.48
ERBB2 P04626 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13915595 0.91 EGFR (0.53) CSF1RNUDT1EGFRERBB2
SCHEMBL13915598 0.86 MAPT (0.51) CSF1R
SCHEMBL2749299 0.86 CSF1R (0.64) CSF1RNUDT1
SCHEMBL5929634 0.83 CSF1R (0.57) CSF1RNUDT1EGFR
SCHEMBL5929704 0.83 CSF1R (0.57) CSF1RNUDT1EGFR
SCHEMBL13915594 0.82 SRC (0.54) EGFRERBB2
SCHEMBL2724559 0.80 CSF1R (0.58) CSF1RNUDT1
SCHEMBL5650362 0.78 ENPP1 (0.55) CSF1REGFR
SCHEMBL12431119 0.78 ENPP1 (0.55) CSF1REGFR
SCHEMBL5929884 0.78 CSF1R (0.56) CSF1RNUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504416-B2 4-substituted quinolines as antitumor agents ASTRAZENECA AB (SE) 2009-03-17 US disclosed
US-7402583-B2 Substituted quinolines as antitumor agents ASTRZENCA AB (SE) 2008-07-22 US disclosed
US-20080027054-A1 4-Substituted quinolines as antitumor agents ASTRAZENECA AB 2008-01-31 US disclosed
US-20070021407-A1 Substituted quinolines as antitumor agents ASTRAZENECA 2007-01-25 US disclosed
US-20070021407-A1 Substituted quinolines as antitumor agents ASTRAZENECA 2007-01-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070021407-A1 Substituted quinolines as antitumor agents NR1H3, NR1H2, NR0B1 CSF1R 182/4885NUDT1 1579/4885EGFR 260/4885
US-20080027054-A1 4-Substituted quinolines as antitumor agents CCNY, TPD52L2, H1-10 CSF1R 991/4885NUDT1 1249/4885EGFR 947/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.