Bambuterol

Bambuterol

SCHEMBL13923751

CN(C)C(=O)Oc1cc(OC(=O)N(C)C)cc([C@@H](O)CNC(C)(C)C)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRB2

The experimentally established mechanism targets of Bambuterol. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADRB2 known ✓ P07550 1/20 1.00
BCHE P06276 6/20 1.00
CYP2D6 P10635 2/20 1.00
ACHE P22303 2/20 1.00
KCNH2 Q12809 1/20 1.00
LMNA P02545 1/20 1.00
CYP2C19 P33261 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bambuterol SCHEMBL4431 1.00 BCHE (1.00) BCHECYP2D6ACHEADRB2KCNH2
Bambuterol SCHEMBL4432 1.00 BCHE (1.00) BCHECYP2D6ACHEADRB2KCNH2
Bambuterol SCHEMBL744580 0.99 BCHE (0.97) BCHECYP2D6ACHEADRB2KCNH2
Bambuterol SCHEMBL1649102 0.97 BCHE (0.95) BCHECYP2D6ACHEADRB2KCNH2
Bambuterol SCHEMBL3713500 0.96 BCHE (0.92) BCHECYP2D6ACHEADRB2KCNH2
SCHEMBL15790253 0.95 BCHE (0.90) BCHECYP2D6ACHEADRB2KCNH2
Bambuterol SCHEMBL21645369 0.95 BCHE (0.90) BCHECYP2D6ACHEADRB2KCNH2
SCHEMBL21674420 0.93 BCHE (0.88) BCHECYP2D6ACHEADRB2KCNH2
Hydrochloric Acid SCHEMBL11123610 0.92 BCHE (0.85) BCHECYP2D6ACHEADRB2KCNH2
SCHEMBL15790471 0.92 BCHE (0.85) BCHECYP2D6ACHEADRB2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115531368-A Application of R-carbamate-beta-phenylethanolamine compounds in treatment of learning and memory deficiency and neurodegenerative diseases 谭文 2022-12-30 CN claimed
WO-2022262873-A2 APPLICATION OF R-CARBAMATE-β-PHENYLETHANOLAMINE COMPOUND IN TREATMENT OF LEARNING AND MEMORY DEFECTS AND NEURODEGENERATIVE DISEASES 谭文 2022-12-22 WO claimed
CN-102448309-A Use of levorotatory bambuterol for the preparation of an inhaled pharmaceutical formulation and combination for the treatment of respiratory disorders WEN TAN 2012-05-09 CN claimed
CN-1638756-A Levo (R) bambuterol and its medicinal use TAN W (ML) 2005-07-13 CN claimed
CN-113613640-B New use of R-enantiomer of adrenergic beta 2 receptor agonist for the treatment of inflammatory bowel disease and parenteral diseases 谭文 2024-11-29 CN disclosed
CN-113613640-B New use of R-enantiomer of adrenergic beta 2 receptor agonist for the treatment of inflammatory bowel disease and parenteral diseases 谭文 2024-11-29 CN disclosed
CN-118787621-A New application of R-salbutamol in treating inflammatory bowel disease and extra-intestinal diseases 谭文 2024-10-18 CN disclosed
EP-4356912-A2 HIGH PENETRATION PRODRUG COMPOSITIONS AND PHARMACEUTICAL COMPOSITION THEREOF FOR TREATMENT OF PULMONARY CONDITIONS Techfields Pharma Co., Ltd. (CN) 2024-04-24 EP disclosed
CN-116077609-B Yellow thick antidiarrheal quick-release pellet for treating IBD and IBS and preparation method thereof 安徽雷允上药业有限公司 2024-04-05 CN disclosed
CN-116077609-A Yellow thick antidiarrheal quick-release pellet for treating IBD and IBS and preparation method thereof 安徽雷允上药业有限公司 2023-05-09 CN disclosed
CN-115531368-A Application of R-carbamate-beta-phenylethanolamine compounds in treatment of learning and memory deficiency and neurodegenerative diseases 谭文 2022-12-30 CN disclosed
CN-115531368-A Application of R-carbamate-beta-phenylethanolamine compounds in treatment of learning and memory deficiency and neurodegenerative diseases 谭文 2022-12-30 CN disclosed
WO-2022262873-A2 APPLICATION OF R-CARBAMATE-β-PHENYLETHANOLAMINE COMPOUND IN TREATMENT OF LEARNING AND MEMORY DEFECTS AND NEURODEGENERATIVE DISEASES 谭文 2022-12-22 WO disclosed
CN-102448309-A Use of levorotatory bambuterol for the preparation of an inhaled pharmaceutical formulation and combination for the treatment of respiratory disorders WEN TAN 2012-05-09 CN disclosed
US-7495028-B2 R-bambuterol, its preparation and therapeutic uses TAN, WEN, DR. 2009-02-24 US disclosed
CN-100356913-C Levo (R) bambuterol and its medicinal use TAN W (CN) 2007-12-26 CN disclosed
CN-1638756-A Levo (R) bambuterol and its medicinal use TAN W (ML) 2005-07-13 CN disclosed