SCHEMBL13925907

SCHEMBL13925907

N#Cc1c(SCC(N)=O)nc(N)c(N)c1-c1ccc(Cl)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.64
ADORA2B P29275 3/20 0.64
ADORA3 P0DMS8 3/20 0.64
ADORA2A P29274 2/20 0.64
ALDH1A1 P00352 8/20 0.61
KDM4E B2RXH2 6/20 0.61
MEN1 O00255 5/20 0.61
KMT2A Q03164 5/20 0.61
HSD17B10 Q99714 5/20 0.61
HPGD P15428 4/20 0.61
ALOX15 P16050 3/20 0.61
MAPT P10636 3/20 0.61
USP2 O75604 1/20 0.61
TP53 P04637 1/20 0.61
L3MBTL1 Q9Y468 1/20 0.61
HTR1B P28222 1/20 0.60
OPRK1 P41145 1/20 0.60
FFAR4 Q5NUL3 1/20 0.60
SIGMAR1 Q99720 1/20 0.60
NPSR1 Q6W5P4 4/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13913699 0.93 ADORA1 (0.72) ADORA1ADORA2BADORA3ADORA2AALDH1A1
SCHEMBL13925701 0.88 ADORA1 (0.64) ADORA1ADORA2BADORA3ADORA2AALDH1A1
SCHEMBL13914100 0.83 ADORA1 (0.76) ADORA1ADORA2BADORA3ADORA2AALDH1A1
SCHEMBL4471026 0.83 ALDH1A1 (0.76) ADORA1ADORA2BADORA3ADORA2AALDH1A1
SCHEMBL13913605 0.82 ADORA1 (0.71) ADORA1ADORA2BADORA3ADORA2AALDH1A1
SCHEMBL13913772 0.82 ALDH1A1 (0.75) ADORA1ADORA2BADORA3ADORA2AALDH1A1
SCHEMBL13913671 0.82 ADORA1 (0.71) ADORA1ADORA2BADORA3ADORA2AALDH1A1
SCHEMBL13914571 0.81 ALDH1A1 (0.65) ADORA1ADORA2BADORA3ADORA2AALDH1A1
SCHEMBL4318226 0.81 ADORA1 (0.70) ADORA1ADORA2BADORA3ADORA2AALDH1A1
SCHEMBL13913704 0.80 ALDH1A1 (0.84) ADORA1ADORA2BADORA3ADORA2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504421-B2 Substituted 2-thio-3,5-dicyano-4-aryl-6-aminopyridines and their use BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-03-17 US disclosed