SCHEMBL13952905

SCHEMBL13952905

CSc1nccc(-c2c3c(C)ccnc3n3c(N)nccc23)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 4/20 0.54
CDK2 P24941 4/20 0.54
CCNA2 P20248 3/20 0.54
CDK5 Q00535 3/20 0.54
CDK5R1 Q15078 3/20 0.54
CCNT1 O60563 2/20 0.54
CCNA1 P78396 2/20 0.54
EPAS1 Q99814 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.37
POLB P06746 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CSNK1E P49674 2/20 0.36
MAPK14 Q16539 3/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
MAPK13 O15264 1/20 0.34
MAPK12 P53778 1/20 0.34
MAPK11 Q15759 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13175411 0.89 CDK9 (0.53) CDK9CDK2CCNA2CDK5CDK5R1
SCHEMBL13175630 0.89 CDK9 (0.55) CDK9CDK2CCNA2CDK5CDK5R1
SCHEMBL13202868 0.87 CDK9 (0.53) CDK9CDK2CCNA2CDK5CDK5R1
SCHEMBL13952907 0.85 CDK2 (0.72) CDK9CDK2CCNA2CDK5CDK5R1
SCHEMBL13952910 0.83 CDK9 (0.56) CDK9CDK2CCNA2CDK5CDK5R1
SCHEMBL13952912 0.81 CDK9 (0.63) CDK9CDK2CCNA2CDK5CDK5R1
SCHEMBL117207 0.81 CDK9 (0.72) CDK9CDK2CCNA2CDK5CDK5R1
SCHEMBL13202831 0.81 CDK9 (0.52) CDK9CDK2CCNA2CDK5CDK5R1
SCHEMBL13220722 0.81 CDK9 (0.57) CDK9CDK2CCNA2CDK5CDK5R1
SCHEMBL14269063 0.80 CDK2 (0.38) CDK9CDK2CCNA2CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7495000-B2 Variolin derivatives and their use as antitumor agents PHARMA MAR, S.A. (ES) 2009-02-24 US disclosed