SCHEMBL13952913

SCHEMBL13952913

CCCCOc1ccnc2c1c(-c1ccnc(OC)n1)c1ccnc(N)n12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 5/20 0.64
CDK5 Q00535 4/20 0.64
CDK5R1 Q15078 4/20 0.64
CDK2 P24941 3/20 0.64
CCNT1 O60563 3/20 0.64
CCNA2 P20248 2/20 0.64
CCNA1 P78396 2/20 0.64
EPAS1 Q99814 1/20 0.36
PDE4B Q07343 1/20 0.33
PDPK1 O15530 1/20 0.32
MAPK13 O15264 1/20 0.31
MAPK12 P53778 1/20 0.31
MAPK11 Q15759 1/20 0.31
MAPK14 Q16539 1/20 0.31
CYP1A2 P05177 2/20 0.31
CYP3A4 P08684 1/20 0.31
TLR8 Q9NR97 3/20 0.31
MCHR1 Q99705 1/20 0.31
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13220724 0.94 CDK9 (0.60) CDK9CDK5CDK5R1CDK2CCNT1
SCHEMBL13220604 0.92 CDK9 (0.58) CDK9CDK5CDK5R1CDK2CCNT1
SCHEMBL13220580 0.89 CDK9 (0.74) CDK9CDK5CDK5R1CDK2CCNT1
SCHEMBL13202878 0.88 CDK9 (0.80) CDK9CDK5CDK5R1CDK2CCNT1
SCHEMBL13952731 0.87 CDK9 (0.59) CDK9CDK5CDK5R1CDK2CCNT1
SCHEMBL13220722 0.85 CDK9 (0.57) CDK9CDK5CDK5R1CDK2CCNT1
SCHEMBL13220539 0.84 CDK9 (0.55) CDK9CDK5CDK5R1CDK2CCNT1
SCHEMBL13202970 0.84 CDK9 (0.61) CDK9CDK5CDK5R1CDK2CCNT1
SCHEMBL13175329 0.82 CDK9 (0.64) CDK9CDK5CDK5R1CDK2CCNT1
SCHEMBL13952912 0.82 CDK9 (0.63) CDK9CDK5CDK5R1CDK2CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7495000-B2 Variolin derivatives and their use as antitumor agents PHARMA MAR, S.A. (ES) 2009-02-24 US disclosed