SCHEMBL13953602

SCHEMBL13953602

C[C@@H](c1ccc(Br)cc1)N1CC[C@](CCN)(c2ccc(F)cc2)OC1=O

nearest known ligand 0.81

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 20/20 0.81
KCNH2 Q12809 1/20 0.79
CYP3A4 P08684 7/20 0.75
CYP2C9 P11712 4/20 0.72
CYP2C19 P33261 3/20 0.68
HSD3B2 P26439 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17120454 0.91 HSD11B1 (0.83) HSD11B1KCNH2CYP3A4CYP2C9CYP2C19
SCHEMBL3638352 0.90 HSD11B1 (1.00) HSD11B1KCNH2CYP3A4CYP2C9CYP2C19
SCHEMBL955653 0.90 HSD11B1 (1.00) HSD11B1KCNH2CYP3A4CYP2C9CYP2C19
SCHEMBL961027 0.90 HSD11B1 (1.00) HSD11B1KCNH2CYP3A4CYP2C9CYP2C19
SCHEMBL955580 0.90 HSD11B1 (1.00) HSD11B1KCNH2CYP3A4CYP2C9CYP2C19
SCHEMBL955578 0.90 HSD11B1 (1.00) HSD11B1KCNH2CYP3A4CYP2C9CYP2C19
SCHEMBL961024 0.90 HSD11B1 (1.00) HSD11B1KCNH2CYP3A4CYP2C9CYP2C19
SCHEMBL955924 0.88 HSD11B1 (1.00) HSD11B1KCNH2CYP3A4CYP2C9CYP2C19
SCHEMBL955921 0.88 HSD11B1 (1.00) HSD11B1KCNH2CYP3A4CYP2C9CYP2C19
SCHEMBL955923 0.88 HSD11B1 (1.00) HSD11B1KCNH2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017664-A1 CYCLIC INHIBITORS OF 11β-HYDROXYSTERIOD DEHYDROGENASE 1 VITAE PHARMACEUTICALS, INC. (US) 2009-02-05 WO disclosed