SCHEMBL13974005

SCHEMBL13974005

CCCc1cccc(-c2nnc(-c3ccc(OC(C)C)c(N)c3)s2)c1CC

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.59
CYP2C9 P11712 5/20 0.45
S1PR3 Q99500 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13974383 0.89 S1PR1 (0.47) S1PR1CYP2C9S1PR3
SCHEMBL12176663 0.81 S1PR1 (0.63) S1PR1S1PR3
SCHEMBL12102768 0.80 S1PR1 (0.59) S1PR1CYP2C9S1PR3
SCHEMBL12176644 0.79 S1PR1 (0.58) S1PR1CYP2C9S1PR3
SCHEMBL12102734 0.78 S1PR1 (0.59) S1PR1S1PR3
SCHEMBL12175246 0.78 S1PR1 (0.61) S1PR1CYP2C9
SCHEMBL12102404 0.77 S1PR1 (0.55) S1PR1CYP2C9S1PR3
SCHEMBL12176643 0.76 S1PR1 (0.46) S1PR1CYP2C9S1PR3
SCHEMBL1293430 0.76 S1PR1 (0.56) S1PR1S1PR3
SCHEMBL2133210 0.74 S1PR1 (1.00) S1PR1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012158550-A2 SELECTIVE HETEROCYCLIC SPHINGOSINE 1 PHOSPHATE RECEPTOR MODULATORS RECEPTOS, INC. (US) 2012-11-22 WO disclosed